Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RTZZCXRVKNMTNQ
|
6.1 | IC50 | 2 | — | |
AQUNLKSSCKKTAO
|
6.1 | IC50 | 2 | — | |
BXKKDJUEVYKLOT
|
6.1 | IC50 | 2 | — | |
GSKXJQZBERQLFV
|
6.1 | IC50 | 2 | — | |
HHRAQYLQCIWYSQ
|
6.1 | IC50 | 2 | — | |
HVFNTCHQZALQNN
|
6.1 | IC50 | 2 | — | |
QSTHQJKUPYALJM
|
6.1 | IC50 | 2 | — | |
STKRPQBTVZSWNF
|
6.1 | IC50 | 2 | — | |
TVDJKFVGGSSMOS
|
6.1 | IC50 | 2 | — | |
ZFUGTFLRENMBAG
|
6.1 | IC50 | 3 | — | |
DNEJKTLTVWWFOX
|
6.1 | IC50 | 2 | — | |
XOMAYDPUCBKVEN
|
6.1 | IC50 | 2 | — | |
NTRNLNAHAHOPNJ
|
6.1 | IC50 | 2 | — | |
JEKLJKGXYFFOIW
|
6.1 | IC50 | 2 | — | |
KAAZDRRTROWGPM
|
6.1 | IC50 | 2 | — | |
OJGUTTIOPDPSMA
|
6.1 | IC50 | 2 | — | |
QWLGKFALYULFFS
|
6.1 | IC50 | 2 | — | |
SCJJJOPARANDTH
|
6.1 | IC50 | 2 | — | |
FSLDLBJGAMZARH
|
6.0 | IC50 | 3 | — | |
JEETZBQOULTRJG
|
6.0 | IC50 | 2 | — | |
JOCCKKDLTYQTDV
|
6.0 | IC50 | 2 | — | |
KTWJPYVRYQJIGD
|
6.0 | IC50 | 2 | — | |
WWKATYZGQPFITE
|
6.0 | IC50 | 2 | — | |
YPNHXGADKUJXJG
|
6.0 | IC50 | 2 | — | |
ZKWJXAYBLHZWQD
|
6.0 | IC50 | 2 | — | |
BFXKLGSNEBEOER
|
6.0 | IC50 | 2 | — | |
LYFSSYUVVYONAT
|
6.0 | IC50 | 2 | — | |
PZWIJHWZZUHCAR
|
6.0 | IC50 | 2 | — | |
ZBODECNZYYNPIT
|
6.0 | IC50 | 2 | — | |
KZOPRHDWMBCDFC
|
6.0 | IC50 | 2 | — | |
LAVMVEIMEUTRHG
|
6.0 | IC50 | 2 | — | |
TXKWHSYYGDZVOC
|
6.0 | IC50 | 2 | — | |
ZSCWIKIEKOGQMJ
|
6.0 | IC50 | 2 | — | |
AGMOZDCBDGTCPZ
|
6.0 | IC50 | 2 | — | |
CXCZBASUFALCKQ
|
6.0 | IC50 | 2 | — | |
DEEQJHMLWWWDLS
|
6.0 | IC50 | 2 | — | |
IZHWKWVIPQQUPL
|
6.0 | IC50 | 2 | — | |
LLUSSJQGFFRYIN
|
6.0 | IC50 | 2 | — | |
MRLPDFXJJBCOPD
|
6.0 | IC50 | 2 | — | |
POCZBHBFCIWCCV
|
6.0 | IC50 | 5 | — | |
QRLIEXSZMDANDN
|
6.0 | IC50 | 2 | — | |
RBJOSAOJJYPLJG
|
6.0 | IC50 | 2 | — | |
RDGSMSLOEKXETJ
|
6.0 | IC50 | 2 | — | |
RHSLCAQORGTADX
|
6.0 | IC50 | 2 | — | |
RMSYQFMJHXZAPA
|
6.0 | Ki | 2 | — | |
SAMSULGCUCSOJQ
|
6.0 | IC50 | 2 | — | |
SHIPZZTUJLMFAJ
|
6.0 | IC50 | 2 | — | |
XRPUJSGGRFQZPJ
|
6.0 | IC50 | 2 | — | |
YXSUPAQPJMXEAF
|
6.0 | IC50 | 2 | — |