Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HISIYDZZYZHWFN
|
6.4 | IC50 | 3 | — | |
JKXYZORDWPTUMV
|
6.4 | IC50 | 2 | — | |
KGERHHFTPBDJEN
|
6.4 | IC50 | 2 | — | |
ZWCPMSLKKDHALP
|
6.4 | IC50 | 2 | — | |
DVSVTNSJQMSOBS
|
6.4 | IC50 | 2 | — | |
FAGVZRREMQKAAQ
|
6.4 | IC50 | 2 | — | |
IKECCCIWJQNGSY
|
6.4 | IC50 | 2 | — | |
BWGHHWSYJIRSQP
|
6.4 | IC50 | 2 | — | |
FRRCHJPQSWYJSH
|
6.4 | IC50 | 4 | — | |
QAQNRWAJNSDKLQ
|
6.4 | IC50 | 2 | — | |
NEVFQPCVHAVFMX
|
6.4 | IC50 | 2 | — | |
WATGOESBZSAATK
|
6.4 | IC50 | 2 | — | |
VOYATJRBIIBIOP
|
6.4 | IC50 | 2 | — | |
AOHAOGINVKWHLM
|
6.4 | IC50 | 2 | — | |
IUUNAOXEWBRZIS
|
6.4 | Ki | 2 | — | |
JMXLXNINVIRWGK
|
6.4 | IC50 | 2 | — | |
UUNOWGXCAZIXDX
|
6.4 | IC50 | 2 | — | |
HGPPRMHXEAZMCS
|
6.4 | IC50 | 3 | — | |
GMYZVEAKJDPVFZ
|
6.3 | IC50 | 2 | — | |
PCIBYKRKILQVKS
|
6.3 | IC50 | 2 | — | |
RFXWTGONAROCHY
|
6.3 | IC50 | 2 | — | |
SAPIEOYWKBEWRF
|
6.3 | IC50 | 2 | — | |
CAZFYBUUYWZTRA
|
6.3 | IC50 | 2 | — | |
NVTRJKGWECZIQW
|
6.3 | IC50 | 2 | — | |
ICQPMQWKTYGPDY
|
6.3 | IC50 | 2 | — | |
PBNNBNYYIVAWGT
|
6.3 | IC50 | 2 | — | |
SLRLQBRWUMWEOZ
|
6.3 | IC50 | 3 | — | |
CTRQACJVRNOHLW
|
6.3 | IC50 | 2 | — | |
ILGVZZSBGPJLHS
|
6.3 | IC50 | 2 | — | |
ITEJDHVEYLBYQP
|
6.3 | IC50 | 2 | — | |
JJGZGELTZPACID
|
6.3 | IC50 | 3 | — | |
KEMCHZMOFUQHQF
|
6.3 | IC50 | 2 | — | |
KNVLMNKVHMDRKF
|
6.3 | IC50 | 2 | — | |
RPFHNYIIVRNCNV
|
6.3 | IC50 | 2 | — | |
VRVGOUHPADQNHC
|
6.3 | IC50 | 2 | — | |
XIFIRTKOEFSDIG
|
6.3 | IC50 | 2 | — | |
YYVXIRSTJYNHFJ
|
6.3 | IC50 | 2 | — | |
ZFQIMJKKFWQMBK
|
6.3 | IC50 | 2 | — | |
AEQWUSSTTYLLFR
|
6.3 | IC50 | 2 | — | |
DMVPQCWNNLBMED
|
6.3 | IC50 | 2 | — | |
NGSHUNXXQUNUDS
|
6.3 | IC50 | 2 | — | |
FGULGOIZBUXLPA
|
6.3 | IC50 | 2 | — | |
FLUZFOGDWLGQJR
|
6.3 | IC50 | 2 | — | |
KCMZLWSTJLSCOT
|
6.3 | IC50 | 2 | — | |
TWUFGLWMAXGSGS
|
6.3 | IC50 | 2 | — | |
ZXYDBRLYEJKZGT
|
6.3 | IC50 | 2 | — | |
IYMHJOBWAFXAAI
|
6.3 | IC50 | 2 | — | |
RDSJPXACTQFSEC
|
6.3 | IC50 | 2 | — | |
AUEORBBRXOLTMO
|
6.3 | IC50 | 2 | — | |
CQJMULDOPNMGJD
|
6.3 | IC50 | 2 | — |