Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DYTQBLYPVPFYLG
|
6.6 | IC50 | 2 | — | |
FPYJSLSYOOTYAQ
|
6.6 | IC50 | 2 | — | |
FTVCCUKUPQHRLI
|
6.6 | IC50 | 2 | — | |
KICKGPQKASOONE
|
6.6 | IC50 | 2 | — | |
MYNDSKARKCPSRA
|
6.6 | IC50 | 2 | — | |
OHHLDOFPDCTGRE
|
6.6 | IC50 | 2 | — | |
PLSLCRVLSLMHSR
|
6.6 | IC50 | 2 | — | |
RVQQPLKLLMDXQS
|
6.6 | IC50 | 2 | — | |
RWYBOYWYRWWRTJ
|
6.6 | IC50 | 2 | — | |
SIPKLTWNJQAWKO
|
6.6 | IC50 | 2 | — | |
YWZPDTMPBUCLEZ
|
6.6 | IC50 | 2 | — | |
QSPZTSNQZUHYRV
|
6.6 | IC50 | 2 | — | |
ABHMLSZZVJVUDO
|
6.6 | IC50 | 2 | — | |
OXVUJFNJJBBQAM
|
6.6 | IC50 | 2 | — | |
BYQMIZKANASQRH
|
6.6 | IC50 | 2 | — | |
JUUCCZVNXSUGRJ
|
6.6 | IC50 | 2 | — | |
XGTWITMCYZSCAI
|
6.6 | IC50 | 2 | — | |
SNMMNXQZLGJXCJ
|
6.6 | IC50 | 2 | — | |
YWZCLODXYXEOJW
|
6.6 | IC50 | 2 | — | |
MIQHJGWVEOELHE
|
6.5 | IC50 | 2 | — | |
UPJZJOAUFLFFAR
|
6.5 | IC50 | 2 | — | |
CTFNTCJGATYTOJ
|
6.5 | IC50 | 2 | — | |
NDWVEFJDUGTQNP
|
6.5 | IC50 | 2 | — | |
ANVMGBJXXQJYER
|
6.5 | IC50 | 2 | — | |
HJESHVHCQSBGRH
|
6.5 | IC50 | 2 | — | |
HLBHMUUNXSMTGA
|
6.5 | IC50 | 2 | — | |
JHZGEAJMTRTONI
|
6.5 | IC50 | 2 | — | |
KMDZXPHEJNVLGD
|
6.5 | IC50 | 2 | — | |
UYLYXNZSRMQYRO
|
6.5 | IC50 | 2 | — | |
CEYVYIFSFUUDBO
|
6.5 | Ki | 2 | — | |
CRYVYILOMSLHLQ
|
6.5 | IC50 | 2 | — | |
GRTMMOOJPZKBCI
|
6.5 | IC50 | 2 | — | |
GYVGQMOJEVZQSW
|
6.5 | IC50 | 2 | — | |
ILQDZDQRPNFMKO
|
6.5 | IC50 | 2 | — | |
QBWLKFUOFUJIPG
|
6.5 | IC50 | 2 | — | |
QDJXHBINRDTWMT
|
6.5 | IC50 | 2 | — | |
HUJPOSGMEWSBGX
|
6.5 | IC50 | 2 | — | |
KHFVQBYEJJEIHG
|
6.5 | IC50 | 2 | — | |
OAWCHZSXBRYHKE
|
6.5 | IC50 | 2 | — | |
YIXSVQYKKJOPJS
|
6.5 | IC50 | 2 | — | |
FWKCJYBRMZTPSS
|
6.5 | IC50 | 2 | — | |
GVGXZBYYIKEWGT
|
6.5 | IC50 | 2 | — | |
ONHNUQYOYCJHED
|
6.5 | IC50 | 2 | — | |
ZFUNYSBCRGYOGS
|
6.5 | IC50 | 2 | — | |
UJQHSSFAJLJAPH
|
6.5 | IC50 | 2 | — | |
BGWWNSJKCPTESJ
|
6.5 | IC50 | 2 | — | |
VRKCLIARHIPPNE
|
6.5 | IC50 | 2 | — | |
XZBREEPFBNJFPK
|
6.5 | IC50 | 2 | — | |
DLKSOJWVTUWOMM
|
6.4 | IC50 | 2 | — | |
FRLMOPXJKYHCTA
|
6.4 | IC50 | 2 | — |