Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TZXRURYHFBZSGH
|
6.8 | Ki | 2 | — | |
YLCZIGRLLGSSOZ
|
6.8 | IC50 | 2 | — | |
GNKSISMYHDFYGM
|
6.8 | IC50 | 2 | — | |
MCPGNKQUPZAGMY
|
6.8 | IC50 | 2 | — | |
OJGJNBQMUGMKTG
|
6.8 | IC50 | 2 | — | |
WPNNXSNEMNITNL
|
6.8 | IC50 | 2 | — | |
JKZBYGUMJOELTM
|
6.8 | IC50 | 2 | — | |
MJWVBEHCIZVLIZ
|
6.8 | IC50 | 2 | — | |
OJPXEBXAMSBWPY
|
6.8 | IC50 | 2 | — | |
PZJGDNRDXHDJEG
|
6.8 | IC50 | 2 | — | |
ZRDTVRVUBKJSLJ
|
6.7 | IC50 | 2 | — | |
GPCMBIWOWUCPEC
|
6.7 | IC50 | 2 | — | |
JDIMCPSYKCGUCK
|
6.7 | IC50 | 2 | — | |
OABQDCYPKAONAC
|
6.7 | IC50 | 2 | — | |
HQAWTGBUKBGURL
|
6.7 | IC50 | 2 | — | |
LRFQYGUWVRUPOU
|
6.7 | IC50 | 2 | — | |
OUVKQCAXDVOIIT
|
6.7 | IC50 | 2 | — | |
ZRVNWWPMGBMFEJ
|
6.7 | IC50 | 2 | — | |
XEJXDTAERYNMJF
|
6.7 | IC50 | 2 | — | |
YYNXNFLCDMNHNK
|
6.7 | IC50 | 2 | — | |
AGZHRZPBUVXTIM
|
6.7 | IC50 | 2 | — | |
AHOZQSJDGWQTGZ
|
6.7 | IC50 | 2 | — | |
ANVMGBJXXQJYER
|
6.7 | IC50 | 2 | — | |
GFAUOHVOSIKURI
|
6.7 | IC50 | 2 | — | |
MUYIQGWTQXWCKY
|
6.7 | IC50 | 2 | — | |
PXMWUCLOPAIDAY
|
6.7 | IC50 | 2 | — | |
QXIWCFSOBHCFPM
|
6.7 | IC50 | 2 | — | |
RUBHAOAJRSDKHD
|
6.7 | IC50 | 2 | — | |
ZTEAMFIIAFKJSO
|
6.7 | IC50 | 2 | — | |
ZYDFILPHGMHKKL
|
6.7 | IC50 | 2 | — | |
WONSGFPKXMEKTD
|
6.7 | IC50 | 2 | — | |
HYNAOOYWCMQTPT
|
6.7 | IC50 | 2 | — | |
SJDBNOPZILRKKB
|
6.7 | IC50 | 2 | — | |
USOOYGCAAUEROH
|
6.7 | IC50 | 2 | — | |
DWJZYCRBKJQBIA
|
6.7 | IC50 | 2 | — | |
DGZYOTRPJLMPMQ
|
6.7 | IC50 | 2 | — | |
DKTKEWPOYRLFDK
|
6.7 | IC50 | 2 | — | |
KPXYCCGYCRCUCJ
|
6.7 | IC50 | 3 | — | |
LTBUMDNUQOPONC
|
6.7 | IC50 | 2 | — | |
VXMMHPAQXRLXQI
|
6.7 | IC50 | 2 | — | |
QYEQAZMKUAVAQT
|
6.7 | IC50 | 2 | — | |
BQKSCZYCLLPPQT
|
6.6 | IC50 | 2 | — | |
IEYXUMXHPMEXLC
|
6.6 | IC50 | 2 | — | |
QCSKEBJTDSIOLJ
|
6.6 | IC50 | 2 | — | |
SGFNNLYTSVJUFM
|
6.6 | IC50 | 2 | — | |
WAAXIFKLWWKGDC
|
6.6 | IC50 | 2 | — | |
HKVHSSSXAMRGND
|
6.6 | IC50 | 2 | — | |
NWBWJYZLVJLKJR
|
6.6 | IC50 | 2 | — | |
ZELHPOQBYBCJFP
|
6.6 | IC50 | 2 | — | |
DWCBYHSUKCYVPJ
|
6.6 | IC50 | 2 | — |