Target Details
| UniProt AC | Q7ZJM1 |
|---|---|
| Gene Symbol | pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 899
- Clinical molecules 0
- Avg pChEMBL 7.3
Active Molecules (899)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXPCMQIDAHRMPC
|
7.0 | IC50 | 2 | — | |
HVDXDXDGCBTPSU
|
6.9 | IC50 | 2 | — | |
NLLFGVOXJVFWDR
|
6.9 | IC50 | 2 | — | |
WJNBDQXVDOJOPE
|
6.9 | IC50 | 2 | — | |
NLGQHMUAHAFRFL
|
6.9 | IC50 | 2 | — | |
CKLUZIMAKNEDFT
|
6.9 | IC50 | 2 | — | |
HDLLPTYGPNZEKD
|
6.9 | IC50 | 2 | — | |
SIUOKPRXJGQHPX
|
6.9 | IC50 | 2 | — | |
ZLOFMAVYNFGKRE
|
6.9 | IC50 | 2 | — | |
JQHRBYOCKAFRDX
|
6.9 | IC50 | 2 | — | |
FWUVZSSWSPORBO
|
6.9 | IC50 | 2 | — | |
DYTGQKUKNHHYRW
|
6.9 | IC50 | 2 | — | |
FIYYRRFBOOVAHE
|
6.9 | IC50 | 2 | — | |
HOODXRHLGKXOKI
|
6.9 | IC50 | 2 | — | |
HXBVMAXHBKSTBQ
|
6.9 | IC50 | 2 | — | |
IEKQWIQTLCCVDM
|
6.9 | IC50 | 2 | — | |
JQTFAOQFMPMHDQ
|
6.9 | IC50 | 2 | — | |
JSKZBUDXJJHWMH
|
6.9 | IC50 | 2 | — | |
KJIZQLFDAULLAK
|
6.9 | IC50 | 2 | — | |
LQEBEYDXCBIMKY
|
6.9 | IC50 | 2 | — | |
NMEFMKZEAMFJPT
|
6.9 | IC50 | 2 | — | |
VLKPQQHJINFIPV
|
6.9 | IC50 | 2 | — | |
VNBMTBOVZFWRAI
|
6.9 | IC50 | 2 | — | |
XGVPVFITNZBZQA
|
6.9 | IC50 | 2 | — | |
XHOFPLVGTCQULP
|
6.9 | IC50 | 2 | — | |
XSRJUIGPNSIGAA
|
6.9 | IC50 | 2 | — | |
ISTSAPNDYCXGDZ
|
6.9 | IC50 | 2 | — | |
BPMDVHPLYAJDGL
|
6.8 | IC50 | 2 | — | |
GSMHULZNHJSXPP
|
6.8 | IC50 | 2 | — | |
JFVFSYGQPDGHQF
|
6.8 | IC50 | 2 | — | |
JVHLCDFNIOKCED
|
6.8 | IC50 | 2 | — | |
KOECUTWWHKLLOJ
|
6.8 | IC50 | 2 | — | |
UXIVWMINNPGARX
|
6.8 | IC50 | 3 | — | |
ZEYRZFOIYUJHEC
|
6.8 | IC50 | 2 | — | |
JJNCAQYXSMGENG
|
6.8 | IC50 | 2 | — | |
FNQPIRNAHZGGGE
|
6.8 | IC50 | 2 | — | |
FZXIXDQTLNIONE
|
6.8 | IC50 | 2 | — | |
UXIVWMINNPGARX
|
6.8 | Kd | 2 | — | |
VZMDZXFRZYBQKO
|
6.8 | IC50 | 2 | — | |
XNPUSRYTYPDIGW
|
6.8 | IC50 | 2 | — | |
GFYGTPODKVZUNL
|
6.8 | IC50 | 2 | — | |
MFNXYTUSFKARCS
|
6.8 | IC50 | 2 | — | |
UQDHFDHSUHECSS
|
6.8 | IC50 | 2 | — | |
VUHPPGIFJGFHHZ
|
6.8 | IC50 | 2 | — | |
CTUQLZDGNOOVRF
|
6.8 | IC50 | 2 | — | |
GGORSCVXKXKHSL
|
6.8 | IC50 | 2 | — | |
JUZRETXRNBMUFO
|
6.8 | IC50 | 2 | — | |
NSURDDQIZZAVJN
|
6.8 | IC50 | 2 | — | |
PJIBKQJSMPMZCH
|
6.8 | IC50 | 3 | — | |
RFVWFGNMGFRBLW
|
6.8 | IC50 | 2 | — |