Target Details
| UniProt AC | Q7Z628 |
|---|---|
| Gene Symbol | NET1 |
| Protein Name | Neuroepithelial cell-transforming gene 1 protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 132
- Clinical molecules 0
- Avg pChEMBL 6.75
Active Molecules (132)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CTYWWUMVNFOYTR
|
6.3 | IC50 | 3 | — | |
UEBNWADIJNYTLV
|
6.3 | IC50 | 3 | — | |
GXDMUUDAPHURSU
|
6.3 | IC50 | 4 | — | |
QIYANFXIRPCCFR
|
6.3 | IC50 | 4 | — | |
WCZIJHPZMNUQAK
|
6.2 | IC50 | 2 | — | |
PCJBHHMLVZKWRN
|
6.2 | IC50 | 3 | — | |
RJMLIMXLXYNFIJ
|
6.2 | IC50 | 3 | — | |
ZQWDWCAENNSUNH
|
6.2 | IC50 | 3 | — | |
WVMDHCAIJWMUKM
|
6.2 | IC50 | 3 | — | |
GWOMMAUEYXPNRP
|
6.2 | IC50 | 2 | — | |
SBKALFWROFTZSP
|
6.1 | IC50 | 2 | — | |
VKXUOQVDGXTZTH
|
6.1 | IC50 | 2 | — | |
HASNBQPSUGYJNL
|
6.1 | IC50 | 3 | — | |
BYXCBFNAGGVRKV
|
6.1 | Ki | 2 | — | |
CIDWBTJORPJQTN
|
6.1 | Ki | 2 | — | |
GLBRSAFDTRHRBW
|
6.1 | IC50 | 3 | — | |
GYNBJBPUCVZGTH
|
6.1 | IC50 | 2 | — | |
LZGLGBOOTDKOQF
|
6.1 | IC50 | 3 | — | |
OKWVFYUPQXMSEV
|
6.1 | IC50 | 2 | — | |
YOVGBLUPSNTJCU
|
6.1 | IC50 | 3 | — | |
KAQUOFCNEYORCQ
|
6.1 | IC50 | 3 | — | |
KAOBGFMQDVKDKV
|
6.1 | IC50 | 2 | — | |
CDXVXAPUCWBZKN
|
6.0 | IC50 | 3 | — | |
NAENGEZVKXADGC
|
6.0 | IC50 | 3 | — | |
JUHSDGAZSHRTAV
|
6.0 | IC50 | 3 | — | |
KPLAPMIQSJDNJP
|
6.0 | IC50 | 3 | — | |
AGRAHYYFJIILCF
|
6.0 | IC50 | 2 | — | |
DFHUUSWJGLRJGV
|
6.0 | IC50 | 3 | — | |
FGAFOULALAFSBX
|
6.0 | IC50 | 2 | — | |
JPPPHDBXUMOMDK
|
6.0 | IC50 | 3 | — | |
POKCWLLPLOIIOW
|
6.0 | IC50 | 3 | — | |
NYDHDNFMMOXOFY
|
6.0 | IC50 | 3 | — |