Target Details
| UniProt AC | Q7Z628 |
|---|---|
| Gene Symbol | NET1 |
| Protein Name | Neuroepithelial cell-transforming gene 1 protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 132
- Clinical molecules 0
- Avg pChEMBL 6.75
Active Molecules (132)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SDFJAHVREUGWBK
|
6.8 | IC50 | 3 | — | |
DIFMRPZOXBYZFC
|
6.8 | IC50 | 3 | — | |
OFNUZQBEAGZOPP
|
6.8 | IC50 | 4 | — | |
MDTFUSLGHFSRLI
|
6.8 | IC50 | 3 | — | |
XNQYQTCZUDFGJQ
|
6.8 | IC50 | 2 | — | |
CIBXZZCJJVKLKR
|
6.7 | IC50 | 3 | — | |
QMMCDRJPRMDPMT
|
6.7 | IC50 | 3 | — | |
FRFZOFGUQVIKSJ
|
6.7 | IC50 | 2 | — | |
XMTSFSJFANMZNO
|
6.7 | IC50 | 3 | — | |
FVPYKEUHDWGTTO
|
6.7 | IC50 | 4 | — | |
KMFJTKOQURPEIV
|
6.7 | IC50 | 3 | — | |
RZJVBWDUILULEO
|
6.7 | IC50 | 2 | — | |
XAXLSVQFDZVYNG
|
6.6 | IC50 | 4 | — | |
YWOVEHIRDVATGZ
|
6.6 | IC50 | 3 | — | |
UCBRSQJQBOWEBP
|
6.6 | IC50 | 3 | — | |
WUZCGLBJMGGJMO
|
6.6 | IC50 | 3 | — | |
QEECCVGAVDCJLV
|
6.6 | IC50 | 2 | — | |
JZYCGFSGFXSIOZ
|
6.6 | IC50 | 3 | — | |
WGNABQIMYMHUQC
|
6.6 | IC50 | 4 | — | |
JTOBXLVKTKGLSL
|
6.6 | IC50 | 4 | — | |
DNTIMCJNBURACB
|
6.5 | IC50 | 3 | — | |
DQKBPLZDDANEEL
|
6.5 | IC50 | 3 | — | |
GHCJADGGBOAAGR
|
6.5 | IC50 | 3 | — | |
TVDNUGUVGACHFB
|
6.5 | IC50 | 4 | — | |
YDGWQVAPZXJCRQ
|
6.5 | IC50 | 3 | — | |
AMKWNLRAFBRBBP
|
6.5 | Ki | 2 | — | |
CIDWBTJORPJQTN
|
6.5 | Ki | 2 | — | |
JUWLARKXKUFQIV
|
6.5 | Ki | 2 | — | |
JUWLARKXKUFQIV
|
6.5 | Ki | 2 | — | |
KNCJEJULKKTIEE
|
6.5 | Ki | 2 | — | |
KNCJEJULKKTIEE
|
6.5 | Ki | 2 | — | |
LZASFPSWSSXPPA
|
6.5 | Ki | 2 | — | |
MENDFCYVYYBFRD
|
6.5 | Ki | 2 | — | |
ROKYHZXDTGMCJT
|
6.5 | Ki | 2 | — | |
ROKYHZXDTGMCJT
|
6.5 | Ki | 2 | — | |
RUZCAHKGJLXNSF
|
6.5 | Ki | 2 | — | |
RXAFOXHLNBBCQQ
|
6.5 | Ki | 2 | — | |
WCUWYYWDWUAFDE
|
6.5 | Ki | 2 | — | |
ZCVHLLHRVFCIKQ
|
6.5 | Ki | 2 | — | |
ZWHDVUZVJSBQRG
|
6.5 | Ki | 2 | — | |
HOXBFDRIDWJAEN
|
6.5 | IC50 | 3 | — | |
CTUZLMXCSKURAB
|
6.5 | IC50 | 2 | — | |
VLARVLVCNCELTO
|
6.5 | IC50 | 2 | — | |
DZUCJYWAUHLCOW
|
6.5 | IC50 | 3 | — | |
XQUUVZDIAMCEHA
|
6.5 | IC50 | 4 | — | |
REVDHAAOZGYXCV
|
6.5 | IC50 | 3 | — | |
DDOQLDAOOODMRN
|
6.4 | IC50 | 3 | — | |
NLISFSAXWFJTGK
|
6.4 | IC50 | 2 | — | |
AMKWNLRAFBRBBP
|
6.3 | Ki | 2 | — | |
SAARGPSTPXUSIL
|
6.3 | IC50 | 4 | — |