Target Details
| UniProt AC | Q7Z628 |
|---|---|
| Gene Symbol | NET1 |
| Protein Name | Neuroepithelial cell-transforming gene 1 protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 132
- Clinical molecules 0
- Avg pChEMBL 6.75
Active Molecules (132)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MSRLFKAAHSYYJT
|
8.4 | IC50 | 4 | — | |
ZXAIYPYVRUXIRT
|
8.2 | IC50 | 3 | — | |
OBWKCACUZGJXHN
|
8.2 | IC50 | 4 | — | |
SWBCLQGKCJMOJJ
|
8.2 | IC50 | 4 | — | |
ZZRHLICOWQQNJL
|
8.1 | IC50 | 4 | — | |
FGMVBSZPVPCFKQ
|
8.0 | IC50 | 4 | — | |
JRSCRGBLGQCTQY
|
7.8 | IC50 | 3 | — | |
LJALDWYVBOLBGW
|
7.7 | IC50 | 4 | — | |
UTQLEVQLADDVHS
|
7.7 | IC50 | 3 | — | |
MKEIWZZHDFWQBD
|
7.7 | IC50 | 4 | — | |
SBZDQHXDTSOYDS
|
7.7 | IC50 | 3 | — | |
FFPZKPBDKMJMOH
|
7.6 | IC50 | 4 | — | |
SYDXJSKTVHXBGQ
|
7.5 | IC50 | 3 | — | |
JLKOYRAHLGKMSS
|
7.5 | IC50 | 3 | — | |
TXLALBNPPFHMQH
|
7.5 | IC50 | 3 | — | |
OISBYAXPTPVNIZ
|
7.5 | IC50 | 3 | — | |
VAXCWNURWRJNKL
|
7.4 | IC50 | 4 | — | |
FNPNFDUAOLYGJY
|
7.4 | IC50 | 3 | — | |
FSYUMFOIUHBSHI
|
7.4 | IC50 | 3 | — | |
QIQXSFJNUMZWBG
|
7.4 | IC50 | 3 | — | |
ADWAGSCYZKTLSE
|
7.3 | IC50 | 3 | — | |
UFFRBOMGNQGCAY
|
7.3 | IC50 | 4 | — | |
YBGWLDSKEUEPKA
|
7.2 | IC50 | 3 | — | |
YBHOJCIKZMRIQL
|
7.2 | IC50 | 3 | — | |
ZJNJPYFFMXVAGY
|
7.2 | IC50 | 4 | — | |
DIOWQSMFSBKMCS
|
7.2 | IC50 | 4 | — | |
PUCWXLYHLYMUCG
|
7.2 | IC50 | 4 | — | |
CLQNHTVQVGGNMJ
|
7.2 | IC50 | 4 | — | |
WDXGJZPPEYWULD
|
7.2 | IC50 | 3 | — | |
ZMQCYFBOOMIJKF
|
7.2 | IC50 | 3 | — | |
MILNRKCCACSUTQ
|
7.1 | IC50 | 3 | — | |
KBCAMMVKABLCAE
|
7.1 | IC50 | 2 | — | |
NDMODESSMWGHBK
|
7.1 | IC50 | 4 | — | |
ROFHPDIVEBIITO
|
7.1 | IC50 | 3 | — | |
LQJSAWJCKIABDN
|
7.1 | IC50 | 3 | — | |
WISXSHNMYCUZHH
|
7.1 | IC50 | 4 | — | |
JKRXUDRMEIXFBV
|
7.0 | IC50 | 4 | — | |
VDPYYIXZGPXIIH
|
7.0 | IC50 | 3 | — | |
CBGYUSPJYFOION
|
7.0 | IC50 | 3 | — | |
QQKNLGCYRCQFQP
|
6.9 | IC50 | 3 | — | |
YVYRBWXITIPQTA
|
6.9 | IC50 | 3 | — | |
IYJBFRBYWMLFEX
|
6.9 | IC50 | 3 | — | |
BCCQIRBEFSTJID
|
6.9 | IC50 | 3 | — | |
SJTJLLXHBQCTJD
|
6.9 | IC50 | 3 | — | |
ZZUJFHUPDOBMOH
|
6.9 | IC50 | 3 | — | |
HSGRXCWTZSFFOF
|
6.9 | IC50 | 3 | — | |
IEEXXKGDHWBIJX
|
6.9 | IC50 | 3 | — | |
FLAQOJMPRHHQFA
|
6.9 | IC50 | 4 | — | |
VIIGZGNGELGDCF
|
6.8 | IC50 | 3 | — | |
YEMZPAKBIRTBDG
|
6.8 | IC50 | 4 | — |