Target Details
| UniProt AC | Q7Z3E1 |
|---|---|
| Gene Symbol | TIPARP |
| Protein Name | Protein mono-ADP-ribosyltransferase TIPARP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) |
Summary
- Multi-target molecules 74
- Clinical molecules 0
- Avg pChEMBL 8.19
Active Molecules (74)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
STSCRAGBCYODMY
|
8.1 | IC50 | 8 | — | |
BMPSOKZAIFFMLK
|
8.1 | IC50 | 6 | — | |
BDQLEBFPVSEZSI
|
8.1 | IC50 | 2 | — | |
MPNZKBPNAZNHSB
|
8.0 | IC50 | 3 | — | |
OORVLKKZQATWIA
|
8.0 | IC50 | 2 | — | |
IESAQQWECFSSTH
|
8.0 | IC50 | 2 | — | |
ZOAMWWAZQUCBSQ
|
8.0 | IC50 | 3 | — | |
GVMXJRXJKMOCBF
|
7.9 | IC50 | 2 | — | |
YUZWVHGUAQAWSV
|
7.9 | IC50 | 2 | — | |
XDYFJQYDGBNPLO
|
7.9 | IC50 | 3 | — | |
TWBMNJILNLYDBC
|
7.8 | IC50 | 3 | — | |
JLVRTMBMCWYGAL
|
7.8 | IC50 | 7 | — | |
SAJUIWASIJXNSM
|
7.7 | IC50 | 2 | — | |
DXFARVNRLJXDDA
|
7.6 | IC50 | 2 | — | |
HISJVPLDLOXJOH
|
7.6 | IC50 | 2 | — | |
YBQAXMUUMRZOKE
|
7.4 | IC50 | 2 | — | |
BOKCRBOZYPDNIC
|
7.4 | IC50 | 3 | — | |
AEOLBQARHQIBTL
|
7.2 | IC50 | 3 | — | |
FSNNMBVVDWKKCB
|
7.1 | IC50 | 6 | — | |
YUBJOUADCHZSHS
|
7.0 | IC50 | 3 | — | |
ACJDTAHNIFCCHB
|
6.8 | IC50 | 3 | — | |
BWTOWBOMDHKCDB
|
6.7 | IC50 | 7 | — | |
MPXAEYSGFKRDQM
|
6.5 | IC50 | 7 | — | |
FDLYAMZZIXQODN
|
6.2 | IC50 | 11 | — |