Target Details
| UniProt AC | Q7Z3E1 |
|---|---|
| Gene Symbol | TIPARP |
| Protein Name | Protein mono-ADP-ribosyltransferase TIPARP |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) |
Summary
- Multi-target molecules 74
- Clinical molecules 0
- Avg pChEMBL 8.19
Active Molecules (74)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WKXCQZQWHUTWSY
|
9.7 | IC50 | 5 | — | |
BAYLVRHCVANSLN
|
9.2 | IC50 | 2 | — | |
BANSZVBMEHYKAV
|
9.2 | IC50 | 4 | — | |
LFYTWGBFZMCREV
|
9.1 | IC50 | 2 | — | |
TWAKELMLSWVDPB
|
8.8 | IC50 | 2 | — | |
LTUOFKFLZDKSRD
|
8.8 | IC50 | 2 | — | |
LBLOWVFFWIQMSQ
|
8.7 | IC50 | 3 | — | |
ZOFBQDSFQVONQL
|
8.7 | IC50 | 2 | — | |
QPPRMYWGJMMFHW
|
8.7 | IC50 | 2 | — | |
LFYTWGBFZMCREV
|
8.7 | IC50 | 2 | — | |
QHKQUHOWXBJVAF
|
8.6 | IC50 | 2 | — | |
SEZOFXSIPYDBSM
|
8.6 | IC50 | 3 | — | |
ZVFTUAXFCXJYHK
|
8.6 | IC50 | 3 | — | |
DKQVFAZKIZXGQF
|
8.6 | IC50 | 2 | — | |
QLYVSWKZQOGBDI
|
8.5 | IC50 | 2 | — | |
BIFMDHUVYGGFCU
|
8.5 | IC50 | 10 | — | |
UQZCQKXJAXKZQH
|
8.5 | IC50 | 4 | — | |
LXMVOWGBBQUTCO
|
8.5 | IC50 | 2 | — | |
WNMYZOLGAGNXGE
|
8.5 | IC50 | 2 | — | |
MJPLTIGFNFYZIV
|
8.5 | IC50 | 2 | — | |
BBLXCPDKVSEZAC
|
8.5 | IC50 | 2 | — | |
JYGANUXFIOAQPJ
|
8.5 | IC50 | 3 | — | |
LBCRVQOCKRRJPU
|
8.5 | IC50 | 2 | — | |
YPLLSXUOZDMWPL
|
8.5 | IC50 | 2 | — | |
ZMNJSCJYCINTTD
|
8.5 | IC50 | 3 | — | |
QRJCYDQKIHFVQC
|
8.4 | IC50 | 3 | — | |
DETVQHYFSHWWBS
|
8.4 | IC50 | 2 | — | |
DETVQHYFSHWWBS
|
8.4 | IC50 | 2 | — | |
LVTXKTNJLIESPY
|
8.4 | IC50 | 2 | — | |
LXMVOWGBBQUTCO
|
8.4 | IC50 | 2 | — | |
QWXXAMNXENCFLM
|
8.4 | IC50 | 2 | — | |
YBQAXMUUMRZOKE
|
8.4 | IC50 | 2 | — | |
LGVKBNNYDKZNJV
|
8.4 | IC50 | 3 | — | |
SAJUIWASIJXNSM
|
8.4 | IC50 | 2 | — | |
CALBKXVDMKLECC
|
8.4 | IC50 | 3 | — | |
IRXHYIYBIYVZMS
|
8.4 | IC50 | 2 | — | |
RQIZHRJCWXOIGA
|
8.4 | IC50 | 2 | — | |
POVGYCDNSJRTOJ
|
8.3 | IC50 | 3 | — | |
ZXYKQNYSXHNQMV
|
8.3 | IC50 | 6 | — | |
BEGHAKMSOKSZMH
|
8.3 | IC50 | 3 | — | |
XFDGHNYVTUXZDC
|
8.3 | IC50 | 2 | — | |
HICODDHJHKXOBW
|
8.3 | IC50 | 2 | — | |
YTQLCJYUTMBQFF
|
8.3 | IC50 | 2 | — | |
DXFARVNRLJXDDA
|
8.3 | IC50 | 2 | — | |
NKUPYUFUIQRZCX
|
8.3 | IC50 | 3 | — | |
VHNNUIFUWOPIHC
|
8.2 | IC50 | 2 | — | |
OIOQXLAIFONXGK
|
8.2 | IC50 | 2 | — | |
NEFFFNZQJIYJPO
|
8.2 | IC50 | 3 | — | |
HICODDHJHKXOBW
|
8.2 | IC50 | 2 | — | |
MJPLTIGFNFYZIV
|
8.2 | IC50 | 2 | — |