Target Details
| UniProt AC | Q7Z2W7 |
|---|---|
| Gene Symbol | TRPM8 |
| Protein Name | Transient receptor potential cation channel subfamily M member 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF18139 (LSDAT_euk) PF25508 (TRPM2) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 6.79
KEGG Pathways (1)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BXXQDSBIEKSNGM
|
8.0 | IC50 | 2 | — | |
ZROLHBHDLIHEMS
|
7.7 | IC50 | 5 | — | |
UQEATFAWAKBMKD
|
7.3 | IC50 | 2 | — | |
QHMBSVQNZZTUGM
|
7.2 | IC50 | 13 | — | |
VUSLIHPWGMCAFY
|
7.2 | IC50 | 2 | — | |
BXXQDSBIEKSNGM
|
7.0 | IC50 | 2 | — | |
UCONUSSAWGCZMV
|
6.8 | IC50 | 4 | — | |
CYQFCXCEBYINGO
|
6.8 | IC50 | 3 | — | |
QXACEHWTBCFNSA
|
6.8 | IC50 | 3 | — | |
SWTFEIIUBMIFPL
|
6.8 | IC50 | 3 | — | |
LEZWWPYKPKIXLL
|
6.4 | IC50 | 20 | — | |
ROGUAPYLUCHQGK
|
6.2 | IC50 | 3 | — | |
HLMBXBGDBBCYII
|
6.1 | IC50 | 3 | — | |
WEWPMAKQEUSKPV
|
6.1 | IC50 | 2 | — | |
REOZWEGFPHTFEI
|
6.0 | IC50 | 4 | — | |
YKPUWZUDDOIDPM
|
6.0 | IC50 | 3 | — |