Target Details
| UniProt AC | Q7X1P7 |
|---|---|
| Gene Symbol | parE |
| Protein Name | DNA topoisomerase (ATP-hydrolyzing) |
| Organism | Streptococcus pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 6.4
Top Co-occurrence Targets
- gyrB 22 shared
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KJDNVMISTFWXEK
|
6.9 | IC50 | 2 | — | |
FQOKIWGLCSLEEB
|
6.8 | IC50 | 2 | — | |
RHKFSMZQNMYMGA
|
6.6 | IC50 | 2 | — | |
FVGMXEKHKSNPMB
|
6.6 | IC50 | 2 | — | |
UTHBRSYQYAZHOI
|
6.6 | IC50 | 2 | — | |
XPIBGMJVUKLMNV
|
6.5 | IC50 | 2 | — | |
CYHRMQQEJPYYQU
|
6.4 | IC50 | 2 | — | |
PRKHQSKTQFWPGJ
|
6.4 | IC50 | 2 | — | |
XMXREKQYAQTQSR
|
6.4 | IC50 | 2 | — | |
PVKBVEDKZQIBPE
|
6.4 | IC50 | 2 | — | |
LXKRVXJCHWCIQA
|
6.4 | IC50 | 2 | — | |
ADEXQHKYMJSASG
|
6.4 | IC50 | 2 | — | |
CXWZHSNLXAJYMQ
|
6.3 | IC50 | 2 | — | |
XGQBLIMXEPFIQW
|
6.3 | IC50 | 2 | — | |
GOCPACVRZTWJMW
|
6.3 | IC50 | 2 | — | |
JUEGEQYABKTKRI
|
6.3 | IC50 | 2 | — | |
WKJAKTPELBFZGV
|
6.2 | IC50 | 2 | — | |
KCCNGWJHGUKZEA
|
6.2 | IC50 | 2 | — | |
QGUJQBAWWLBPDZ
|
6.2 | IC50 | 2 | — | |
ULDPAUYYMDRQGQ
|
6.2 | IC50 | 2 | — | |
OIKPUVGIFBCWLO
|
6.1 | IC50 | 2 | — | |
LPYHBQXASYFYSZ
|
6.0 | IC50 | 2 | — |