Target Details
| UniProt AC | Q7L7X3 |
|---|---|
| Gene Symbol | TAOK1 |
| Protein Name | Serine/threonine-protein kinase TAO1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 179
- Clinical molecules 27
- Avg pChEMBL 6.64
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (179)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XOOAAYRIVATZNM
|
6.2 | Ki | 55 | — | |
ZCCJKVBTHCOISJ
|
6.2 | Ki | 46 | — | |
AQKQATGZIKRZMQ
|
6.1 | Ki | 16 | — | |
BIIVYFLTOXDAOV
|
6.1 | Ki | 31 | — | |
BLQYVHBZHAISJM
|
6.1 | Ki | 54 | — | |
JTRNNNVASYCTLO
|
6.1 | Ki | 14 | — | |
LJKJYKWDLJUZHA
|
6.1 | Ki | 24 | — | |
MCKPYPWHBUXLEZ
|
6.1 | Ki | 21 | — | |
OUSFTKFNBAZUKL
|
6.1 | Ki | 58 | Yes | |
RWEHAHIEUDLKGT
|
6.1 | Ki | 33 | — | |
STUPRWVTVIXNLF
|
6.1 | Ki | 6 | — | |
VCFDMLBPASGZTP
|
6.1 | Ki | 38 | — | |
XBYVOPRDASFDMY
|
6.1 | Ki | 42 | — | |
ZXLFIHLBHMLHFJ
|
6.1 | Ki | 31 | — | |
VAARYSWULJUGST
|
6.1 | Kd | 119 | Yes | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes | |
BPNUQXPIQBZCMR
|
6.0 | Ki | 60 | — | |
CLRFYTGANQZOBS
|
6.0 | Ki | 41 | — | |
GXJSLIOOPZRPEV
|
6.0 | Ki | 34 | — | |
HKZKELVPGXJIMW
|
6.0 | Ki | 41 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KBFBKKNSHPUFET
|
6.0 | Ki | 5 | — | |
KLZLCOULUPUMAI
|
6.0 | Ki | 3 | — | |
MHWHPWMWKYXCRJ
|
6.0 | Ki | 32 | — | |
RJZDECGDCKOHBV
|
6.0 | Ki | 70 | — | |
SPMHGQZFMNZCBV
|
6.0 | Ki | 30 | Yes | |
UCLBDUZAAUTHBW
|
6.0 | Ki | 4 | — | |
WAKGEHXTOOFEAE
|
6.0 | Ki | 27 | — | |
ZBNZXTGUTAYRHI
|
6.0 | Ki | 102 | Yes |