Target Details
| UniProt AC | Q7L7X3 |
|---|---|
| Gene Symbol | TAOK1 |
| Protein Name | Serine/threonine-protein kinase TAO1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 179
- Clinical molecules 27
- Avg pChEMBL 6.64
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (179)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SFPWNTQWFFNJIH
|
6.4 | Ki | 48 | — | |
URNZTLZSAVLTIZ
|
6.4 | Ki | 26 | — | |
XMGFTZYNTYNOOJ
|
6.4 | Ki | 10 | — | |
VOQXQYXTZZHYBF
|
6.4 | IC50 | 7 | Yes | |
OYONTEXKYJZFHA
|
6.3 | Kd | 69 | Yes | |
BPNUQXPIQBZCMR
|
6.3 | Kd | 83 | Yes | |
UJIAQDJKSXQLIT
|
6.3 | Kd | 38 | — | |
AILRADAXUVEEIR
|
6.3 | IC50 | 75 | — | |
CODOEMQMKTTYRW
|
6.3 | IC50 | 7 | — | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — | |
AHJRHEGDXFFMBM
|
6.3 | Ki | 28 | — | |
BLXRLDWQFVTLLB
|
6.3 | IC50 | 2 | — | |
BVNBRKOALNETGX
|
6.3 | IC50 | 2 | — | |
CTALVCVKEYVQIJ
|
6.3 | IC50 | 2 | — | |
CTTLBTOARINAOQ
|
6.3 | IC50 | 2 | — | |
DZSUJUOJJJCWGG
|
6.3 | Ki | 55 | Yes | |
FEWKYLIQAFEHAS
|
6.3 | IC50 | 2 | — | |
FUMCKNCUEAQHCV
|
6.3 | Ki | 103 | — | |
HRZOUBQYVUXBNS
|
6.3 | Ki | 38 | — | |
JJJSCYSPSKBQAX
|
6.3 | Ki | 34 | — | |
KYAGDWQXJICEFO
|
6.3 | IC50 | 2 | — | |
LCGSWTFWYNYUKS
|
6.3 | Ki | 26 | — | |
MBGWYGHZHAXUFZ
|
6.3 | IC50 | 2 | — | |
MKUQVFUKAUXYEW
|
6.3 | IC50 | 2 | — | |
MLHQXLYJVYMVNC
|
6.3 | IC50 | 2 | — | |
NLUPJKQOKWBWFC
|
6.3 | Ki | 69 | — | |
NWRZXVYYHQMCAU
|
6.3 | IC50 | 2 | — | |
OIEFVAVADRALOZ
|
6.3 | IC50 | 2 | — | |
OWDRQHVEJIYVOI
|
6.3 | Ki | 47 | — | |
QSAYKRXJXDKAIM
|
6.3 | IC50 | 2 | — | |
QTLUCZVJQWOZNL
|
6.3 | IC50 | 2 | — | |
UBIKJGRVXIINFB
|
6.3 | IC50 | 2 | — | |
UKZSZOYTVQHXML
|
6.3 | IC50 | 2 | — | |
UXGKCQZWBHGMBU
|
6.3 | IC50 | 2 | — | |
VCKRURAVBSHCHK
|
6.3 | IC50 | 2 | — | |
ZEGLWOVBWQUGAL
|
6.3 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
6.3 | Kd | 85 | Yes | |
CHQYAWLKOUOTQO
|
6.2 | IC50 | 20 | — | |
JRNJNYBQQYBCLE
|
6.2 | Kd | 40 | Yes | |
KGPGFQWBCSZGEL
|
6.2 | Kd | 59 | Yes | |
CHTMRWQLNNRRFJ
|
6.2 | Ki | 70 | — | |
GEGCXGMFUYJULA
|
6.2 | Ki | 30 | Yes | |
HFNKQEVNSGCOJV
|
6.2 | Ki | 18 | — | |
KEZAHTDTAWUZDU
|
6.2 | Ki | 8 | — | |
LRINYHMQZRENCY
|
6.2 | Ki | 29 | — | |
PCQMERRARZKTPW
|
6.2 | Ki | 68 | — | |
RTDSHUGNRVXRHN
|
6.2 | Ki | 51 | — | |
VSVWQTDDGQSGHP
|
6.2 | Ki | 51 | — | |
WPHKIQPVPYJNAX
|
6.2 | Ki | 81 | — | |
XHORJSJFHVABEA
|
6.2 | Ki | 49 | — |