Target Details
| UniProt AC | Q7L7X3 |
|---|---|
| Gene Symbol | TAOK1 |
| Protein Name | Serine/threonine-protein kinase TAO1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 179
- Clinical molecules 27
- Avg pChEMBL 6.64
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (179)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKLPOUDFRUNULX
|
6.8 | IC50 | 2 | — | |
JRVGQZOVEXJARK
|
6.8 | IC50 | 2 | — | |
JSGUDZBCODXIII
|
6.8 | IC50 | 2 | — | |
MJXKBVJFXOMGJZ
|
6.8 | IC50 | 2 | — | |
MLYQDOZQEYXGTC
|
6.8 | IC50 | 2 | — | |
OZYLOBCEPYGHNK
|
6.8 | IC50 | 2 | — | |
QLJIETHEHOPBEV
|
6.8 | IC50 | 2 | — | |
QLWPBOYRMFPURQ
|
6.8 | IC50 | 2 | — | |
SEVCBWKJSOLMNQ
|
6.8 | Ki | 38 | — | |
XJSFDMGICAWQFS
|
6.8 | Ki | 60 | — | |
YEHCNYAQEBQCCS
|
6.8 | Ki | 74 | — | |
ZAGFGDPXBTWJKY
|
6.8 | IC50 | 2 | — | |
ZKPHMJAXPXACLF
|
6.8 | IC50 | 2 | — | |
ZVWRFVCNQOECJS
|
6.8 | Ki | 71 | — | |
ZZSRKSMPHPUYRC
|
6.8 | IC50 | 2 | — | |
YRDHKIFCGOZTGD
|
6.8 | IC50 | 21 | — | |
LGHBDVLAHHANMX
|
6.7 | Ki | 53 | — | |
MZDKLVOWGIOKTN
|
6.7 | Ki | 80 | — | |
NRGYZNJPCGRCLV
|
6.7 | Ki | 52 | — | |
XCHWBXBDZRJVDP
|
6.7 | Ki | 51 | — | |
VKBFHTIUXUCYRQ
|
6.7 | Ki | 66 | — | |
RZUOCXOYPYGSKL
|
6.6 | Kd | 8 | — | |
CUIHSIWYWATEQL
|
6.6 | Kd | 61 | Yes | |
FLEAYYMORDPWAJ
|
6.6 | Ki | 90 | — | |
JPCWMTOYDYYXLS
|
6.6 | Ki | 7 | — | |
LYNBNVBMAGDJRW
|
6.6 | Ki | 81 | — | |
NWAUBAGBGOPJLF
|
6.6 | Ki | 51 | Yes | |
NWMPVMMGSHXANZ
|
6.6 | Ki | 58 | — | |
PTVPBWWDGZSEAF
|
6.6 | Ki | 63 | — | |
RKUKAACYUCUJEE
|
6.6 | Ki | 58 | — | |
XKZQZMSAWVDRSP
|
6.6 | Ki | 39 | Yes | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
ADMFLILDQJSEIK
|
6.5 | Ki | 72 | — | |
AIQDZMUPVYDVLB
|
6.5 | Ki | 48 | — | |
GNLAGGCSJGJECE
|
6.5 | Ki | 19 | Yes | |
HXHAJRMTJXHJJZ
|
6.5 | Ki | 52 | Yes | |
MPVGZUGXCQEXTM
|
6.5 | Kd | 61 | Yes | |
NFMGZVPRGVERNN
|
6.5 | Ki | 44 | — | |
NJPWCTYVEJIQBM
|
6.5 | Ki | 72 | — | |
RTYJMUXLFRYRBU
|
6.5 | Ki | 35 | — | |
UJBJWYNPUOLFIZ
|
6.5 | Ki | 49 | — | |
XBAIEEJJCJHBDL
|
6.5 | Ki | 17 | — | |
XFWUTMHVDGPWLH
|
6.5 | Ki | 75 | — | |
XTVULKIROSNNTG
|
6.5 | Ki | 29 | — | |
KSERXGMCDHOLSS
|
6.4 | Kd | 3 | — | |
KNACLJBHKVSTDL
|
6.4 | Ki | 40 | — | |
MQRDVGBWWVWMEN
|
6.4 | Ki | 47 | — | |
NKEUPUJTVALZIK
|
6.4 | Ki | 28 | — | |
RGNHKJWHFIPHIM
|
6.4 | Ki | 66 | — | |
SDBOIBYRBWPIEL
|
6.4 | Ki | 31 | — |