Target Details
| UniProt AC | Q7L7X3 |
|---|---|
| Gene Symbol | TAOK1 |
| Protein Name | Serine/threonine-protein kinase TAO1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 179
- Clinical molecules 27
- Avg pChEMBL 6.64
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (179)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
QDITZBLZQQZVEE
|
8.7 | Kd | 19 | — | |
IFPPYSWJNWHOLQ
|
8.2 | Ki | 52 | Yes | |
HKSZLNNOFSGOKW
|
8.0 | Ki | 118 | — | |
MWKSRKSEWLRPBL
|
7.9 | Kd | 1075 | — | |
OSVUGUHRKMMBSE
|
7.8 | Kd | 170 | — | |
SRUYMJRFVGLQDV
|
7.8 | Ki | 37 | — | |
DKZYXHCYPUVGAF
|
7.8 | Kd | 112 | — | |
DGLFSNZWRYADFC
|
7.7 | IC50 | 12 | — | |
DSSNAGYVGTYAGH
|
7.7 | IC50 | 10 | — | |
MVJMMLFMPWITEJ
|
7.7 | Ki | 110 | — | |
IXLOPQOCFOQEQN
|
7.6 | Ki | 2 | — | |
KDKUVYLMPJIGKA
|
7.6 | Ki | 91 | Yes | |
NXSJMRCTGYTSTK
|
7.6 | Kd | 200 | — | |
OWRXHGAFWZFFCW
|
7.6 | Ki | 113 | — | |
QQWUGDVOUVUTOY
|
7.6 | Kd | 231 | Yes | |
ODPGGGTTYSGTGO
|
7.5 | Kd | 153 | — | |
UMTWTCVTRDYHQQ
|
7.5 | Ki | 56 | — | |
BMIWGAPTSPJEJO
|
7.3 | IC50 | 2 | — | |
CHEWOUMVNNRPQL
|
7.3 | IC50 | 2 | — | |
CMHKKTGCFWZUEZ
|
7.3 | IC50 | 2 | — | |
HWNWXVSQBFOHFT
|
7.3 | IC50 | 2 | — | |
IWFBETHWIWFHFI
|
7.3 | IC50 | 2 | — | |
JZZXFSWUEYNLNZ
|
7.3 | IC50 | 2 | — | |
LYJAJWGXMOKLOA
|
7.3 | IC50 | 2 | — | |
SEJNBCOCDTVEAV
|
7.3 | IC50 | 2 | — | |
USKFTJSEVSYZHZ
|
7.3 | IC50 | 2 | — | |
YBMXZSWZDVESLG
|
7.3 | IC50 | 2 | — | |
OLVBAUVSICCWEJ
|
7.2 | Ki | 39 | — | |
PROLIXHVRCJEFH
|
7.2 | Ki | 46 | — | |
SACRIVBWIXWZAH
|
7.2 | Ki | 4 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
GCBJDOWIQHMCMR
|
7.1 | Ki | 84 | — | |
WFTZMAAMCVPJJT
|
7.1 | Ki | 26 | — | |
MCCCQFAOMZMZKE
|
7.0 | Ki | 52 | — | |
RYYNGWLOYLRZLK
|
7.0 | Ki | 104 | — | |
ULHGAQSVFPOUDY
|
7.0 | Ki | 43 | — | |
YMIJUBCSOKSFRU
|
7.0 | Ki | 87 | — | |
UZWDCWONPYILKI
|
7.0 | Kd | 47 | — | |
BSFNGHCTZDCQBF
|
6.9 | Ki | 93 | — | |
GSXRCPJTNIGKSZ
|
6.9 | Ki | 43 | — | |
KUNZDWIFPOMUOX
|
6.9 | Ki | 36 | — | |
TVUWQDLBEOZVOU
|
6.9 | Ki | 41 | — | |
MFAQYJIYDMLAIM
|
6.9 | Kd | 130 | Yes | |
OVPNQJVDAFNBDN
|
6.9 | Kd | 44 | Yes | |
BIIVYFLTOXDAOV
|
6.8 | Kd | 82 | Yes | |
KTEIFNKAUNYNJU
|
6.8 | Ki | 48 | — | |
AJLWHEZEVCJFTK
|
6.8 | IC50 | 2 | — | |
CVJUGGSXRCYDMH
|
6.8 | IC50 | 2 | — | |
DKSNLQYRZJKYOC
|
6.8 | Ki | 51 | — |