Target Details
| UniProt AC | Q7KZI7 |
|---|---|
| Gene Symbol | MARK2 |
| Protein Name | Serine/threonine-protein kinase MARK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 133
- Clinical molecules 16
- Avg pChEMBL 6.68
Associated Diseases (1)
Active Molecules (133)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NLUPJKQOKWBWFC
|
6.2 | Ki | 69 | — | |
RYAVJHIPOWNWDE
|
6.2 | Ki | 38 | — | |
UJLAWZDWDVHWOW
|
6.2 | Ki | 11 | — | |
XBYVOPRDASFDMY
|
6.2 | Ki | 42 | — | |
ZRQXCQXWTLVASO
|
6.2 | Ki | 36 | — | |
HFNKQEVNSGCOJV
|
6.2 | Kd | 65 | — | |
KOZFSFOOLUUIGY
|
6.2 | Kd | 88 | Yes | |
KGPGFQWBCSZGEL
|
6.1 | Kd | 59 | Yes | |
IZAVTOABECKIDH
|
6.1 | Ki | 20 | — | |
MQRDVGBWWVWMEN
|
6.1 | Ki | 47 | — | |
NHFDRBXTEDBWCZ
|
6.1 | Ki | 41 | — | |
NRGYZNJPCGRCLV
|
6.1 | Ki | 52 | — | |
NRZYTPAJGVTKIM
|
6.1 | Ki | 38 | — | |
OADRBDVURCEKRP
|
6.1 | Ki | 44 | — | |
PUPCRRRSBUYJAD
|
6.1 | Ki | 44 | Yes | |
UGEJLCNSVIVALC
|
6.1 | Ki | 41 | — | |
XSRHBCYNCKAFKS
|
6.1 | Ki | 45 | — | |
YEHCNYAQEBQCCS
|
6.1 | Ki | 74 | — | |
GCIKSSRWRFVXBI
|
6.0 | Ki | 109 | Yes | |
GHPFQRTVUDXWCC
|
6.0 | Ki | 35 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JAMDNXUAYUHJLJ
|
6.0 | Ki | 40 | — | |
JSDGKSMNPHJDFK
|
6.0 | Ki | 35 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KNACLJBHKVSTDL
|
6.0 | Ki | 40 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NWAUBAGBGOPJLF
|
6.0 | Ki | 51 | Yes | |
QQUXFYAWXPMDOE
|
6.0 | Ki | 31 | — | |
SEVCBWKJSOLMNQ
|
6.0 | Ki | 38 | — | |
SFPWNTQWFFNJIH
|
6.0 | Ki | 48 | — | |
ULHGAQSVFPOUDY
|
6.0 | Ki | 43 | — | |
XAYDUCQADQTDGX
|
6.0 | Ki | 12 | — | |
XYXLUJQBBIBJFV
|
6.0 | Ki | 36 | — |