Target Details
| UniProt AC | Q79MP6 |
|---|---|
| Gene Symbol | blaIMP-1 |
| Protein Name | Beta-lactamase |
| Organism | Pseudomonas aeruginosa |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00753 (Lactamase_B) |
Summary
- Multi-target molecules 219
- Clinical molecules 0
- Avg pChEMBL 8.23
Top Co-occurrence Targets
- blaNDM-1 203 shared
- vim-1 202 shared
- blaVIM-2 194 shared
- 15 shared
- bla(tem-2) 1 shared
- tem-1 1 shared
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZFMNMVNGJGVQRC
|
10.3 | IC50 | 4 | — | |
QMSLEPRJPQOPQL
|
10.0 | IC50 | 4 | — | |
RODLLQWLAUOVIQ
|
9.9 | IC50 | 4 | — | |
RXVDHGMURRZHLL
|
9.9 | IC50 | 4 | — | |
JHKJCVLYLVBLCQ
|
9.9 | IC50 | 4 | — | |
CAYHAEYZSNEDCI
|
9.8 | IC50 | 4 | — | |
AADKYZQKXNREKK
|
9.7 | IC50 | 4 | — | |
GKMVNXKFFZYSNJ
|
9.7 | IC50 | 4 | — | |
FFRWLTARAWFRFC
|
9.6 | IC50 | 4 | — | |
GGUJAXXOLRPBFQ
|
9.6 | IC50 | 4 | — | |
OULGJNXHRCRUSI
|
9.6 | IC50 | 4 | — | |
HZGTYRHUZKQSRT
|
9.6 | IC50 | 4 | — | |
FZNMIJSHTQATBE
|
9.6 | IC50 | 4 | — | |
DKIUQWRXQIXNFD
|
9.5 | IC50 | 4 | — | |
IZHRFZDSEMSKQW
|
9.4 | IC50 | 4 | — | |
LBOBSCGMRITHQL
|
9.4 | IC50 | 4 | — | |
IZRGISIZXAAYTN
|
9.4 | IC50 | 4 | — | |
JAUOOHBTAFQCND
|
9.4 | IC50 | 4 | — | |
MWJSNGDGUXWXJE
|
9.3 | IC50 | 4 | — | |
NSEYRXDYYZWBRO
|
9.3 | IC50 | 4 | — | |
UEUUAQDRRFZXAD
|
9.3 | IC50 | 4 | — | |
JVBIDFOKKKQDHM
|
9.3 | IC50 | 4 | — | |
LYQXKOGPSMULQJ
|
9.3 | IC50 | 4 | — | |
IKLQJYOBZMJSDZ
|
9.3 | IC50 | 4 | — | |
QLFCRTVWKSWUJV
|
9.3 | IC50 | 4 | — | |
KBXJSJVSIFCCMH
|
9.3 | IC50 | 4 | — | |
GSOMLHAHEABUCB
|
9.2 | IC50 | 4 | — | |
JTPLYTQKVPUMTN
|
9.2 | IC50 | 4 | — | |
LSDLDSCILQRABC
|
9.2 | IC50 | 4 | — | |
XCECLESCRLJFHL
|
9.2 | IC50 | 4 | — | |
DJDJBTVGPINQTN
|
9.2 | IC50 | 4 | — | |
CLUGWDOUECRLLK
|
9.2 | IC50 | 4 | — | |
WGNFSUAOZYDIRY
|
9.2 | IC50 | 4 | — | |
AVFNAPQOQDOLRK
|
9.2 | IC50 | 4 | — | |
FQFYCZPTOXFNDS
|
9.2 | IC50 | 4 | — | |
UNMZOEHSYGRTHM
|
9.2 | IC50 | 4 | — | |
FRABTOZORWZALU
|
9.1 | IC50 | 4 | — | |
VPMZIWLEJLBHHN
|
9.1 | IC50 | 4 | — | |
GEFNYGUKJDHWHO
|
9.1 | IC50 | 4 | — | |
HLOVJTXLVHNCDN
|
9.1 | IC50 | 4 | — | |
WQFKQLWLEFFNKQ
|
9.1 | IC50 | 4 | — | |
PNVQTEQVHFQOLJ
|
9.1 | IC50 | 4 | — | |
LYQXKOGPSMULQJ
|
9.0 | IC50 | 4 | — | |
BYIRAZZBHXLXQG
|
9.0 | IC50 | 4 | — | |
QDRNELLVCKPVOG
|
9.0 | IC50 | 4 | — | |
ODGLPRDZERDAQX
|
8.9 | IC50 | 4 | — | |
XHDVBGDIWMBBAX
|
8.9 | IC50 | 4 | — | |
KHOHRDFIYPATSQ
|
8.9 | IC50 | 4 | — | |
QZPAESVLFNOPHO
|
8.9 | IC50 | 4 | — | |
YBLPXPGATOTWRZ
|
8.9 | IC50 | 4 | — |