Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MMQKXGDYQHMHSZ
|
7.5 | IC50 | 2 | — | |
OZYHJYRSCKCZKX
|
7.5 | IC50 | 2 | — | |
STFNWTMRBYIMLT
|
7.5 | IC50 | 2 | — | |
FTAFMNFWYJKAJJ
|
7.5 | IC50 | 2 | — | |
KCYXSYRXHHMSBC
|
7.5 | IC50 | 2 | — | |
QWEZWEWKCUNZJG
|
7.5 | IC50 | 2 | — | |
MKBOLWCAEVSPDO
|
7.5 | IC50 | 2 | — | |
UDKLDLMPRXYJPF
|
7.5 | IC50 | 2 | — | |
UWKBMEKSJZFOCU
|
7.5 | IC50 | 2 | — | |
VQKRGMYOAWQGCE
|
7.5 | IC50 | 2 | — | |
ZOHLWPAZJWTAHT
|
7.5 | IC50 | 2 | — | |
IECKFYAGOUPMJR
|
7.4 | IC50 | 2 | — | |
JOMOIXVBAURLGQ
|
7.4 | IC50 | 2 | — | |
SGHKDINHXLFACS
|
7.4 | IC50 | 2 | — | |
BAPPEEFNOHFHHS
|
7.4 | IC50 | 2 | — | |
PPCMZJZCQJICAL
|
7.4 | IC50 | 2 | — | |
UHKGVUWBDHSDRE
|
7.4 | IC50 | 2 | — | |
YUKIZQHXWJBIDQ
|
7.4 | IC50 | 2 | — | |
AWHRLSWFNXNGCA
|
7.4 | IC50 | 2 | — | |
CVCIBCNUVGMNFI
|
7.4 | IC50 | 2 | — | |
FIZLYPSCDVIWPS
|
7.4 | IC50 | 2 | — | |
FWUVZSSWSPORBO
|
7.4 | IC50 | 2 | — | |
GTEGUHHUOZACRM
|
7.4 | IC50 | 2 | — | |
JKMGFMMJBBZMJM
|
7.4 | IC50 | 2 | — | |
KOIRVGGHXVYBOP
|
7.4 | IC50 | 2 | — | |
LQRHHCHTXASMRR
|
7.4 | IC50 | 2 | — | |
NBZUOYQZKBUFGU
|
7.4 | IC50 | 2 | — | |
NNXBNFFXSZUCOX
|
7.4 | IC50 | 2 | — | |
NOODFABEYJETRJ
|
7.4 | IC50 | 2 | — | |
PAGOKHJLPJSOGR
|
7.4 | Ki | 2 | — | |
QQDBOQBXQGDIRP
|
7.4 | IC50 | 2 | — | |
UTWNIOAXAGJMTO
|
7.4 | IC50 | 2 | — | |
VPLYPNIQVTUPJL
|
7.4 | IC50 | 2 | — | |
WWUWVEGTBIZBFG
|
7.4 | IC50 | 2 | — | |
VLKPQQHJINFIPV
|
7.4 | IC50 | 2 | — | |
WBSJEVXLQLNTQL
|
7.4 | IC50 | 2 | — | |
DKFIIFFRTUHRER
|
7.4 | IC50 | 2 | — | |
NHVRMORBBFOPFV
|
7.4 | IC50 | 2 | — | |
SYXPFHAWSHIXAB
|
7.4 | IC50 | 2 | — | |
DFLZMXAKNICYGN
|
7.4 | IC50 | 2 | — | |
IVCJOZWNBVIQMX
|
7.4 | IC50 | 2 | — | |
VACAAOPFMOFFDX
|
7.4 | IC50 | 2 | — | |
NNCDBLPXXVWRGR
|
7.4 | IC50 | 2 | — | |
UKWKHQJMIGMBTM
|
7.4 | IC50 | 2 | — | |
MDXLFERPCWCEQE
|
7.3 | IC50 | 2 | — | |
OSYORQDUUBUZPF
|
7.3 | IC50 | 2 | — | |
VFRFSNWOJFIQFA
|
7.3 | IC50 | 2 | — | |
XEYPVNLDIUAZEN
|
7.3 | IC50 | 2 | — | |
NABWPXICBAZTPN
|
7.3 | IC50 | 2 | — | |
QDZYVQLHEZVPBI
|
7.3 | IC50 | 2 | — |