Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IQEXWNMHBMERCT
|
7.7 | IC50 | 2 | — | |
FXOSOEDOGWALNW
|
7.6 | IC50 | 2 | — | |
IGVFBVBNNDZUPO
|
7.6 | IC50 | 2 | — | |
JOIBXXXZWAARGO
|
7.6 | IC50 | 2 | — | |
MBSMKNIEBKYDJI
|
7.6 | IC50 | 3 | — | |
IFEXVYKQUYKHHL
|
7.6 | IC50 | 2 | — | |
NYTDLCMIWTXHQU
|
7.6 | IC50 | 2 | — | |
RJRJCEILQXCOQW
|
7.6 | IC50 | 2 | — | |
WWPKBJCPIBCDLA
|
7.6 | IC50 | 2 | — | |
XIPCSYYWFBSFKD
|
7.6 | IC50 | 2 | — | |
YZIAZOQBKIGPGH
|
7.6 | IC50 | 2 | — | |
DRDHSNVHWKKIHX
|
7.6 | IC50 | 2 | — | |
MABLQILTRUMWKO
|
7.6 | IC50 | 2 | — | |
NBJWZVPLWARKGD
|
7.6 | IC50 | 2 | — | |
GOAIEZIUJNGELQ
|
7.6 | IC50 | 2 | — | |
IGPCYZSJTNKDBD
|
7.6 | IC50 | 2 | — | |
YSIMBNDIQQVRNI
|
7.6 | IC50 | 2 | — | |
DALAMXZEIWIEOM
|
7.6 | IC50 | 2 | — | |
ZMWNOXHZOQBNOQ
|
7.6 | IC50 | 2 | — | |
WXIZJLLJYKSHOJ
|
7.6 | IC50 | 2 | — | |
KVDQIQQSORQTEK
|
7.5 | IC50 | 2 | — | |
RJWBOLLTMJMYNV
|
7.5 | IC50 | 2 | — | |
SFDWYBWLCUHBOM
|
7.5 | IC50 | 2 | — | |
CXSATMSLNBALME
|
7.5 | IC50 | 2 | — | |
CYJVKJHOTQQQQB
|
7.5 | IC50 | 2 | — | |
DQJCPBNTEWWPSV
|
7.5 | IC50 | 2 | — | |
HPKRJZKNJPQFCU
|
7.5 | IC50 | 2 | — | |
LOZAOFDCUDUZNL
|
7.5 | IC50 | 2 | — | |
MWPWGZXQCAMTQA
|
7.5 | IC50 | 3 | — | |
NPQLJDQNIHSLCI
|
7.5 | IC50 | 2 | — | |
OLEQHARKFQIMPD
|
7.5 | IC50 | 2 | — | |
OVFCNJTZFINERB
|
7.5 | IC50 | 2 | — | |
SWTCOVTZHCWWLN
|
7.5 | IC50 | 2 | — | |
SYXMVDKLNDHJCN
|
7.5 | IC50 | 2 | — | |
TYJVGQMIOMQMDL
|
7.5 | IC50 | 2 | — | |
YCHXPKWHIKUTAJ
|
7.5 | IC50 | 2 | — | |
YWFVTSHPZBFEBT
|
7.5 | IC50 | 2 | — | |
ZMNBZCGHGFFNNU
|
7.5 | IC50 | 2 | — | |
HVWVEBJNUHGACI
|
7.5 | IC50 | 2 | — | |
KNXSVCHOFRTUQC
|
7.5 | IC50 | 2 | — | |
OHSMGUZDDMBFSC
|
7.5 | IC50 | 2 | — | |
CGRYPFQLSPYBQD
|
7.5 | IC50 | 2 | — | |
FLTRTAWGZZZNLI
|
7.5 | IC50 | 2 | — | |
HDXMXTOTDSAUFD
|
7.5 | IC50 | 2 | — | |
OJSHOMJTWMYBRH
|
7.5 | IC50 | 2 | — | |
UWBJMUHRCSGGGI
|
7.5 | IC50 | 2 | — | |
AGPDHYVMIWYSBH
|
7.5 | IC50 | 3 | — | |
HDYOIHVTWSZHQB
|
7.5 | IC50 | 2 | — | |
JQDYJMIGQQKXRD
|
7.5 | IC50 | 2 | — | |
MMNYINTURABQHM
|
7.5 | IC50 | 2 | — |