Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGLXZAUYBWNGQB
|
8.1 | IC50 | 2 | — | |
LQCPHYOUQIUBMP
|
8.1 | IC50 | 2 | — | |
PRHMKGKKUARNFW
|
8.1 | IC50 | 2 | — | |
QYFLJDZFSUYSQK
|
8.1 | IC50 | 2 | — | |
SPQKOMZYUIKCAR
|
8.1 | IC50 | 2 | — | |
TZMIHRDKFQXCPK
|
8.1 | IC50 | 2 | — | |
UOFGXMDVJQLSIB
|
8.1 | IC50 | 2 | — | |
VQKMITXYEKFPGK
|
8.1 | IC50 | 2 | — | |
XFUNUTLEVXBIFL
|
8.1 | IC50 | 2 | — | |
YZYLVRWBRSZBRJ
|
8.1 | IC50 | 2 | — | |
ZSDBGBUACZIEEL
|
8.1 | IC50 | 2 | — | |
CILGSVOXLMYHRS
|
8.0 | IC50 | 2 | — | |
KKDNFRLOMQTWSZ
|
8.0 | IC50 | 2 | — | |
SIDXJUHOOIRQED
|
8.0 | IC50 | 2 | — | |
XRNBUPRKOYQWFN
|
8.0 | IC50 | 2 | — | |
CURDSQDCFXPHFD
|
8.0 | IC50 | 2 | — | |
BAPPEEFNOHFHHS
|
8.0 | IC50 | 2 | — | |
BKHJHHIIMXQCTK
|
8.0 | IC50 | 2 | — | |
BYWWWBVBUHYGJN
|
8.0 | IC50 | 2 | — | |
CBSXIVIKLPREOK
|
8.0 | IC50 | 2 | — | |
FSMARROOKZZWJX
|
8.0 | IC50 | 2 | — | |
FTYLDFCKUWPBJJ
|
8.0 | IC50 | 2 | — | |
FWWMQCWKOSWTOL
|
8.0 | IC50 | 2 | — | |
FYXXIVCLXLOWRN
|
8.0 | IC50 | 3 | — | |
GPFNPLCMOSSWHU
|
8.0 | IC50 | 2 | — | |
IZXCRCGHEJFQPK
|
8.0 | IC50 | 2 | — | |
JFNWNZHZNZMNAC
|
8.0 | IC50 | 2 | — | |
JKWMCNLVARUYBJ
|
8.0 | IC50 | 2 | — | |
JYELQJPRWOTTBL
|
8.0 | IC50 | 2 | — | |
KBXRRIUYQIDSON
|
8.0 | IC50 | 2 | — | |
MBAXAWROWFFEGK
|
8.0 | IC50 | 2 | — | |
MNBWNMFAAQFCNB
|
8.0 | IC50 | 2 | — | |
OKLYWXAJDGCACQ
|
8.0 | IC50 | 4 | — | |
PSMBVVQBAVEJQO
|
8.0 | IC50 | 2 | — | |
QBJQWIQAJVYVTJ
|
8.0 | IC50 | 2 | — | |
RWCACWKLMSUOFC
|
8.0 | IC50 | 2 | — | |
SLWYUJVCKLWTGV
|
8.0 | IC50 | 2 | — | |
TWWLJWGXKQAITK
|
8.0 | IC50 | 2 | — | |
UJZVTGOPYAKBIB
|
8.0 | IC50 | 2 | — | |
UMPCIKHDGHZMJR
|
8.0 | IC50 | 2 | — | |
XWVTVSSPEHHYCE
|
8.0 | IC50 | 2 | — | |
YLSDEWQNSIAMQO
|
8.0 | IC50 | 3 | — | |
YMHFTOMTCCFRNK
|
8.0 | IC50 | 2 | — | |
YWYHIDAJZXGQKF
|
8.0 | IC50 | 2 | — | |
ZEVLDMFFBCKSHX
|
8.0 | IC50 | 2 | — | |
ZUIYPJQQZGBVLU
|
8.0 | IC50 | 2 | — | |
BWVZWKYMWWPRBX
|
8.0 | IC50 | 2 | — | |
KYHZUFQVCKRYFE
|
8.0 | IC50 | 2 | — | |
QAWUWJFJRCHDON
|
8.0 | IC50 | 2 | — | |
QOZUICSVLJMIDW
|
8.0 | IC50 | 2 | — |