Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GRTMMOOJPZKBCI
|
6.5 | IC50 | 2 | — | |
GYVGQMOJEVZQSW
|
6.5 | IC50 | 2 | — | |
ILQDZDQRPNFMKO
|
6.5 | IC50 | 2 | — | |
QBWLKFUOFUJIPG
|
6.5 | IC50 | 2 | — | |
QDJXHBINRDTWMT
|
6.5 | IC50 | 2 | — | |
KHFVQBYEJJEIHG
|
6.5 | IC50 | 2 | — | |
OAWCHZSXBRYHKE
|
6.5 | IC50 | 2 | — | |
FWKCJYBRMZTPSS
|
6.5 | IC50 | 2 | — | |
HUJPOSGMEWSBGX
|
6.5 | IC50 | 2 | — | |
YIXSVQYKKJOPJS
|
6.5 | IC50 | 2 | — | |
GVGXZBYYIKEWGT
|
6.5 | IC50 | 2 | — | |
ILVWSEURLCBURN
|
6.5 | IC50 | 2 | — | |
UJQHSSFAJLJAPH
|
6.5 | IC50 | 2 | — | |
VFQDFESUBBNARZ
|
6.5 | IC50 | 2 | — | |
BGWWNSJKCPTESJ
|
6.5 | IC50 | 2 | — | |
VRKCLIARHIPPNE
|
6.5 | IC50 | 2 | — | |
XZBREEPFBNJFPK
|
6.5 | IC50 | 2 | — | |
DLKSOJWVTUWOMM
|
6.4 | IC50 | 2 | — | |
JKXYZORDWPTUMV
|
6.4 | IC50 | 2 | — | |
KGERHHFTPBDJEN
|
6.4 | IC50 | 2 | — | |
RMPNLEUIIWOMGN
|
6.4 | IC50 | 2 | — | |
ZWCPMSLKKDHALP
|
6.4 | IC50 | 2 | — | |
DVSVTNSJQMSOBS
|
6.4 | IC50 | 2 | — | |
FAGVZRREMQKAAQ
|
6.4 | IC50 | 2 | — | |
IKECCCIWJQNGSY
|
6.4 | IC50 | 2 | — | |
BWGHHWSYJIRSQP
|
6.4 | IC50 | 2 | — | |
FRRCHJPQSWYJSH
|
6.4 | IC50 | 4 | — | |
QAQNRWAJNSDKLQ
|
6.4 | IC50 | 2 | — | |
NEVFQPCVHAVFMX
|
6.4 | IC50 | 2 | — | |
WATGOESBZSAATK
|
6.4 | IC50 | 2 | — | |
VOYATJRBIIBIOP
|
6.4 | IC50 | 2 | — | |
IUUNAOXEWBRZIS
|
6.4 | Ki | 2 | — | |
JMXLXNINVIRWGK
|
6.4 | IC50 | 2 | — | |
UUNOWGXCAZIXDX
|
6.4 | IC50 | 2 | — | |
HGPPRMHXEAZMCS
|
6.4 | IC50 | 3 | — | |
GMYZVEAKJDPVFZ
|
6.3 | IC50 | 2 | — | |
PCIBYKRKILQVKS
|
6.3 | IC50 | 2 | — | |
RFXWTGONAROCHY
|
6.3 | IC50 | 2 | — | |
SAPIEOYWKBEWRF
|
6.3 | IC50 | 2 | — | |
ICQPMQWKTYGPDY
|
6.3 | IC50 | 2 | — | |
PBNNBNYYIVAWGT
|
6.3 | IC50 | 2 | — | |
CTRQACJVRNOHLW
|
6.3 | IC50 | 2 | — | |
ILGVZZSBGPJLHS
|
6.3 | IC50 | 2 | — | |
LDKJJCMTYSYKGC
|
6.3 | IC50 | 2 | — | |
ITEJDHVEYLBYQP
|
6.3 | IC50 | 2 | — | |
JJGZGELTZPACID
|
6.3 | IC50 | 3 | — | |
KEMCHZMOFUQHQF
|
6.3 | IC50 | 2 | — | |
KNVLMNKVHMDRKF
|
6.3 | IC50 | 2 | — | |
RPFHNYIIVRNCNV
|
6.3 | IC50 | 2 | — | |
VRVGOUHPADQNHC
|
6.3 | IC50 | 2 | — |