Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZYDFILPHGMHKKL
|
6.7 | IC50 | 2 | — | |
WONSGFPKXMEKTD
|
6.7 | IC50 | 2 | — | |
HYNAOOYWCMQTPT
|
6.7 | IC50 | 2 | — | |
SJDBNOPZILRKKB
|
6.7 | IC50 | 2 | — | |
USOOYGCAAUEROH
|
6.7 | IC50 | 2 | — | |
DWJZYCRBKJQBIA
|
6.7 | IC50 | 2 | — | |
DGZYOTRPJLMPMQ
|
6.7 | IC50 | 2 | — | |
DKTKEWPOYRLFDK
|
6.7 | IC50 | 2 | — | |
KPXYCCGYCRCUCJ
|
6.7 | IC50 | 3 | — | |
LTBUMDNUQOPONC
|
6.7 | IC50 | 2 | — | |
VXMMHPAQXRLXQI
|
6.7 | IC50 | 2 | — | |
QYEQAZMKUAVAQT
|
6.7 | IC50 | 2 | — | |
IEYXUMXHPMEXLC
|
6.6 | IC50 | 2 | — | |
QCSKEBJTDSIOLJ
|
6.6 | IC50 | 2 | — | |
SGFNNLYTSVJUFM
|
6.6 | IC50 | 2 | — | |
WAAXIFKLWWKGDC
|
6.6 | IC50 | 2 | — | |
AAYAGLDVWRKOPN
|
6.6 | IC50 | 2 | — | |
HKVHSSSXAMRGND
|
6.6 | IC50 | 2 | — | |
NWBWJYZLVJLKJR
|
6.6 | IC50 | 2 | — | |
DWCBYHSUKCYVPJ
|
6.6 | IC50 | 2 | — | |
DYTQBLYPVPFYLG
|
6.6 | IC50 | 2 | — | |
FPYJSLSYOOTYAQ
|
6.6 | IC50 | 2 | — | |
FTVCCUKUPQHRLI
|
6.6 | IC50 | 2 | — | |
MYNDSKARKCPSRA
|
6.6 | IC50 | 2 | — | |
OHHLDOFPDCTGRE
|
6.6 | IC50 | 2 | — | |
PLSLCRVLSLMHSR
|
6.6 | IC50 | 2 | — | |
QSPZTSNQZUHYRV
|
6.6 | IC50 | 2 | — | |
RVQQPLKLLMDXQS
|
6.6 | IC50 | 2 | — | |
RWYBOYWYRWWRTJ
|
6.6 | IC50 | 2 | — | |
SIPKLTWNJQAWKO
|
6.6 | IC50 | 2 | — | |
YWZPDTMPBUCLEZ
|
6.6 | IC50 | 2 | — | |
ZELHPOQBYBCJFP
|
6.6 | IC50 | 2 | — | |
ABHMLSZZVJVUDO
|
6.6 | IC50 | 2 | — | |
BYQMIZKANASQRH
|
6.6 | IC50 | 2 | — | |
JUUCCZVNXSUGRJ
|
6.6 | IC50 | 2 | — | |
XGTWITMCYZSCAI
|
6.6 | IC50 | 2 | — | |
SNMMNXQZLGJXCJ
|
6.6 | IC50 | 2 | — | |
YWZCLODXYXEOJW
|
6.6 | IC50 | 2 | — | |
MIQHJGWVEOELHE
|
6.5 | IC50 | 2 | — | |
UPJZJOAUFLFFAR
|
6.5 | IC50 | 2 | — | |
CTFNTCJGATYTOJ
|
6.5 | IC50 | 2 | — | |
NDWVEFJDUGTQNP
|
6.5 | IC50 | 2 | — | |
ANVMGBJXXQJYER
|
6.5 | IC50 | 2 | — | |
HJESHVHCQSBGRH
|
6.5 | IC50 | 2 | — | |
HLBHMUUNXSMTGA
|
6.5 | IC50 | 2 | — | |
JHZGEAJMTRTONI
|
6.5 | IC50 | 2 | — | |
KMDZXPHEJNVLGD
|
6.5 | IC50 | 2 | — | |
UYLYXNZSRMQYRO
|
6.5 | IC50 | 2 | — | |
CEYVYIFSFUUDBO
|
6.5 | Ki | 2 | — | |
CRYVYILOMSLHLQ
|
6.5 | IC50 | 2 | — |