Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NQHLSBKNTGZGQE
|
7.0 | IC50 | 2 | — | |
ROIUPYVFSXZOEO
|
7.0 | IC50 | 2 | — | |
ROWZYDNMRQHGQR
|
7.0 | IC50 | 2 | — | |
TZXRURYHFBZSGH
|
7.0 | Ki | 2 | — | |
XTPXVUSZRLMULQ
|
7.0 | IC50 | 2 | — | |
YXIMJFMQWKJZCT
|
7.0 | IC50 | 2 | — | |
ATDMGAIFDCLGGH
|
7.0 | IC50 | 2 | — | |
HHOMTASMRVIHQK
|
7.0 | IC50 | 2 | — | |
FNUPPEQQWCCTQZ
|
7.0 | IC50 | 2 | — | |
VEXNNTLYFREDFU
|
7.0 | IC50 | 3 | — | |
BMKDHJRRYRCOJM
|
7.0 | IC50 | 2 | — | |
IVERODHAYRWQDN
|
7.0 | IC50 | 2 | — | |
SDBYEHYJCQSIJI
|
7.0 | IC50 | 2 | — | |
VWBPLONFZAKNAY
|
7.0 | IC50 | 2 | — | |
YNKQBPAMXZCFHI
|
7.0 | IC50 | 2 | — | |
QUDSBEUEJPRFOE
|
7.0 | IC50 | 2 | — | |
CMMROMAIEJESHS
|
7.0 | IC50 | 2 | — | |
DWGMJZOSEGIGHX
|
7.0 | IC50 | 2 | — | |
GUPBCFZJCLSQGL
|
7.0 | IC50 | 2 | — | |
HJVVPRFMGAXBBU
|
7.0 | IC50 | 2 | — | |
IQVWIKWYURRSAA
|
7.0 | IC50 | 2 | — | |
KPSUATBRKZSLGB
|
7.0 | IC50 | 2 | — | |
OCYCJENTLYSSKA
|
7.0 | IC50 | 2 | — | |
VBGFNEQSLWFVHW
|
7.0 | IC50 | 2 | — | |
WYJIXJFPLGPWKT
|
7.0 | IC50 | 2 | — | |
ZJNVQCQCAACIOY
|
7.0 | IC50 | 2 | — | |
IKBRTKBQTBPMJM
|
7.0 | IC50 | 2 | — | |
KBIRJUUJIOKTBK
|
7.0 | IC50 | 2 | — | |
AVEADFUBEJNYMC
|
7.0 | IC50 | 2 | — | |
FVNBSBGNENHAFN
|
7.0 | IC50 | 2 | — | |
KTMKXZDZXDYLAP
|
7.0 | IC50 | 2 | — | |
KTMKXZDZXDYLAP
|
7.0 | IC50 | 2 | — | |
LNOZHNZDRONKFT
|
7.0 | IC50 | 2 | — | |
LWPSCCFYFDSPEC
|
7.0 | IC50 | 2 | — | |
NDRTUAJATMBOBN
|
7.0 | IC50 | 2 | — | |
NIYSFVZEKVNKDE
|
7.0 | IC50 | 2 | — | |
SDUJKGMHVYFQHR
|
7.0 | IC50 | 2 | — | |
YWZSBKOZYMDNCK
|
7.0 | IC50 | 2 | — | |
ZXPCMQIDAHRMPC
|
7.0 | IC50 | 2 | — | |
HVDXDXDGCBTPSU
|
6.9 | IC50 | 2 | — | |
NLLFGVOXJVFWDR
|
6.9 | IC50 | 2 | — | |
WJNBDQXVDOJOPE
|
6.9 | IC50 | 2 | — | |
NLGQHMUAHAFRFL
|
6.9 | IC50 | 2 | — | |
CKLUZIMAKNEDFT
|
6.9 | IC50 | 2 | — | |
GEAUCNNPRRTTJD
|
6.9 | IC50 | 2 | — | |
HDLLPTYGPNZEKD
|
6.9 | IC50 | 2 | — | |
SIUOKPRXJGQHPX
|
6.9 | IC50 | 2 | — | |
ZLOFMAVYNFGKRE
|
6.9 | IC50 | 2 | — | |
JQHRBYOCKAFRDX
|
6.9 | IC50 | 2 | — | |
GSMHULZNHJSXPP
|
6.9 | IC50 | 2 | — |