Target Details
| UniProt AC | Q76353 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00665 (rve) |
Summary
- Multi-target molecules 806
- Clinical molecules 0
- Avg pChEMBL 7.29
Active Molecules (806)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
INDBQLZJXZLFIT
|
9.7 | IC50 | 5 | — | |
WHTVZRBIWZFKQO
|
9.6 | IC50 | 4 | — | |
IJMJMINUWKUWGH
|
9.1 | IC50 | 2 | — | |
KAUSSVRICVWZOF
|
9.0 | IC50 | 2 | — | |
IJMJMINUWKUWGH
|
9.0 | IC50 | 2 | — | |
FUAAWFQZWQTORD
|
8.7 | IC50 | 2 | — | |
GOXOIUKALCKLBR
|
8.7 | IC50 | 2 | — | |
JRJOAWBBGFRSKN
|
8.7 | IC50 | 2 | — | |
OHEKQGOBJIKKIF
|
8.7 | IC50 | 2 | — | |
SZMXBVLFEKAFCW
|
8.7 | IC50 | 2 | — | |
UQNGYUIYLKHANY
|
8.7 | IC50 | 2 | — | |
RHWKPHLQXYSBKR
|
8.6 | IC50 | 2 | — | |
BLAAHOHPTRRHEE
|
8.5 | IC50 | 2 | — | |
GJVSFGHPHYFQLR
|
8.5 | IC50 | 2 | — | |
HFZMUFCMKBURCR
|
8.5 | IC50 | 2 | — | |
IDFBTAAZGBQVFK
|
8.5 | IC50 | 2 | — | |
JDRPVKFHRSSYPE
|
8.5 | IC50 | 2 | — | |
MWOWPHYFPJLZBJ
|
8.5 | IC50 | 2 | — | |
PEUHOTMXYZUPRW
|
8.5 | IC50 | 2 | — | |
PYYHHGCMPCSNFK
|
8.5 | IC50 | 2 | — | |
RRWKTKIOQUKLPC
|
8.5 | IC50 | 2 | — | |
SHVZIYWVYKHZTQ
|
8.5 | IC50 | 2 | — | |
UMJDGJBTISXJDU
|
8.5 | IC50 | 2 | — | |
WCWSTNLSLKSJPK
|
8.5 | IC50 | 2 | — | |
WSDGRLFPCSFYMS
|
8.5 | IC50 | 2 | — | |
CBTMLQQUKGUWIY
|
8.4 | IC50 | 2 | — | |
CEHXEXNUZXZFBO
|
8.4 | IC50 | 2 | — | |
DVTZVOHNHIDPQF
|
8.4 | IC50 | 2 | — | |
FQNCLQBMLDMZCA
|
8.4 | IC50 | 2 | — | |
GPUWROATNJMQHS
|
8.4 | IC50 | 2 | — | |
GTWKEOPOJIKGNC
|
8.4 | IC50 | 2 | — | |
GXQOKLJRGLAGLA
|
8.4 | IC50 | 2 | — | |
HWPPBTBVGPCSCA
|
8.4 | IC50 | 2 | — | |
NDYNDZNHTYFBJC
|
8.4 | IC50 | 2 | — | |
NFEPQYVYHPMREC
|
8.4 | IC50 | 2 | — | |
NKASXVZVFGZXDX
|
8.4 | IC50 | 2 | — | |
PEUHOTMXYZUPRW
|
8.4 | IC50 | 2 | — | |
PYZPPVJYQJWLSA
|
8.4 | IC50 | 2 | — | |
UYQJZKVDHPVDOB
|
8.4 | IC50 | 2 | — | |
WALXSGFVDFDFRD
|
8.4 | IC50 | 2 | — | |
YFSHCUFOGWJTAO
|
8.4 | IC50 | 2 | — | |
ZNALLTSSUXRQGH
|
8.4 | IC50 | 2 | — | |
KKDNFRLOMQTWSZ
|
8.4 | IC50 | 2 | — | |
HHTJOARSCIPIIU
|
8.4 | IC50 | 2 | — | |
YGAWXQMGZYJGAP
|
8.4 | IC50 | 2 | — | |
CDKMAVRQWDOIFA
|
8.3 | IC50 | 2 | — | |
ADDAVDPIWMAUCW
|
8.3 | IC50 | 2 | — | |
AOIQERYGVZXFRM
|
8.3 | IC50 | 2 | — | |
BKXKYZADTBYFKB
|
8.3 | IC50 | 2 | — | |
BRUIGFVBEPZHAV
|
8.3 | IC50 | 2 | — |