Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DSLRRJIAXNZCSG
|
7.7 | IC50 | 2 | — | |
HGABZLMUWONTSR
|
7.7 | IC50 | 2 | — | |
ISHYYUYNFLXJQS
|
7.7 | IC50 | 2 | — | |
NUELOPFROCIPLJ
|
7.7 | IC50 | 2 | — | |
QLLSKLPCLTYSAW
|
7.7 | IC50 | 2 | — | |
WKCGEYBYESUICW
|
7.7 | IC50 | 2 | — | |
CQFUGLCPSNTKAO
|
7.7 | IC50 | 2 | — | |
GEAUCNNPRRTTJD
|
7.7 | IC50 | 2 | — | |
GXWODWMYKXULHQ
|
7.7 | IC50 | 3 | — | |
MJMDFEZUPZGSHT
|
7.7 | IC50 | 2 | — | |
UNPFEEFPHCXQCF
|
7.7 | IC50 | 2 | — | |
WOULWISOHTZRJX
|
7.7 | IC50 | 2 | — | |
YIBOMRUWOWDFLG
|
7.7 | IC50 | 6 | — | |
MHUVLRNBDLFMHQ
|
7.7 | IC50 | 2 | — | |
RUMMDAPDDLJACC
|
7.7 | IC50 | 2 | — | |
ZSYYYYOMVLMTCF
|
7.7 | Ki | 2 | — | |
BTKYDHWMZTUHMW
|
7.6 | IC50 | 2 | — | |
GCEGOTUYYWDPTF
|
7.6 | IC50 | 2 | — | |
IYYSVJVCUFTVLZ
|
7.6 | IC50 | 2 | — | |
JAPBEUUVCDEABS
|
7.6 | IC50 | 2 | — | |
KYDALGOIRAPGOG
|
7.6 | IC50 | 2 | — | |
LKDMBBITLLHPTI
|
7.6 | IC50 | 2 | — | |
LYSDBGPVDHWBSR
|
7.6 | IC50 | 2 | — | |
MEFZDWSXKDPPAP
|
7.6 | IC50 | 2 | — | |
NIFNGKZDXZYIAL
|
7.6 | IC50 | 2 | — | |
OHNFSFKNDCPQPZ
|
7.6 | IC50 | 2 | — | |
RMPNLEUIIWOMGN
|
7.6 | IC50 | 2 | — | |
UVHPTIHVNPHEKS
|
7.6 | IC50 | 2 | — | |
UXDWYQAXEGVSPS
|
7.6 | IC50 | 3 | — | |
XPCJVVJMITVUDR
|
7.6 | IC50 | 2 | — | |
YHRQSPRSRROVMC
|
7.6 | IC50 | 2 | — | |
VQWNFBGVGJSEIS
|
7.6 | IC50 | 3 | — | |
FHEIBFFRHYMBMZ
|
7.6 | IC50 | 2 | — | |
GHQLRJSTAXRERC
|
7.6 | IC50 | 2 | — | |
GZMNOTZGPCNHSP
|
7.6 | IC50 | 2 | — | |
IVPUMMMSBHDOHK
|
7.6 | IC50 | 2 | — | |
JLHZDKWPASMSGJ
|
7.6 | IC50 | 2 | — | |
LFMGOGFQQXQENP
|
7.6 | IC50 | 2 | — | |
NFTOJSQFJKWPBJ
|
7.6 | IC50 | 2 | — | |
NMTZHGMDHMNRSK
|
7.6 | IC50 | 2 | — | |
PNHXTVWKZGVUSJ
|
7.6 | IC50 | 2 | — | |
QBMNFDFNTDZHAM
|
7.6 | IC50 | 2 | — | |
QWCPXRJTQSFQIA
|
7.6 | IC50 | 2 | — | |
VJQXBJRSFHAPJG
|
7.6 | IC50 | 2 | — | |
VRKMJGDGFOBMKJ
|
7.6 | IC50 | 2 | — | |
VYQAEVMCBBKRGE
|
7.6 | IC50 | 2 | — | |
XHNLVFGRVFKGSQ
|
7.6 | IC50 | 2 | — | |
DTHZUSMREBJMBT
|
7.6 | IC50 | 2 | — | |
FESKECLMGVLGFJ
|
7.6 | IC50 | 2 | — | |
AGHMFOBRJGGWOS
|
7.6 | IC50 | 2 | — |