Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PQHZDLWZDBGFLW
|
7.8 | IC50 | 2 | — | |
QVDWPWSANSQTHD
|
7.8 | IC50 | 2 | — | |
TXUZIUVPQOEQIE
|
7.8 | IC50 | 2 | — | |
UIMJDZAUFISWPN
|
7.8 | IC50 | 2 | — | |
CPIULLPZAYZFJW
|
7.7 | IC50 | 2 | — | |
DTZKZNPNNCEVDZ
|
7.7 | IC50 | 2 | — | |
XHGMYKUMNYJNAH
|
7.7 | IC50 | 2 | — | |
GKJQZUMJYPWMMQ
|
7.7 | IC50 | 2 | — | |
DFGPETMJUAEASQ
|
7.7 | IC50 | 2 | — | |
GQMQZXHAMCLBEK
|
7.7 | IC50 | 2 | — | |
JNCKVSZNUFQNSW
|
7.7 | IC50 | 2 | — | |
KHGOZPBXQQRDPS
|
7.7 | IC50 | 2 | — | |
KJQMIGLUMAJBDG
|
7.7 | IC50 | 2 | — | |
LQBLCVLTPIUNBP
|
7.7 | IC50 | 2 | — | |
MORWDLWHAAPLCE
|
7.7 | IC50 | 2 | — | |
NDOMDMSDXSLLHI
|
7.7 | IC50 | 2 | — | |
OSNHXMBZJPUQKF
|
7.7 | IC50 | 2 | — | |
PYWHKNREYNCJNZ
|
7.7 | IC50 | 2 | — | |
UFZKXRFAXDLHOV
|
7.7 | IC50 | 2 | — | |
ZQCPKQJODQWPGV
|
7.7 | IC50 | 2 | — | |
HIDJVTANKWMNAG
|
7.7 | IC50 | 2 | — | |
MJLVOIVXLAWOLL
|
7.7 | IC50 | 2 | — | |
AHAQASQWEHMCHG
|
7.7 | IC50 | 2 | — | |
ALKIIYOVOOKGCB
|
7.7 | IC50 | 2 | — | |
BJJHNPCGDRJFQW
|
7.7 | IC50 | 2 | — | |
CGPUDIUUVSBGLW
|
7.7 | IC50 | 2 | — | |
GLQCTOKPQDLBOJ
|
7.7 | IC50 | 2 | — | |
GLXUBTVPJONLFB
|
7.7 | IC50 | 2 | — | |
JCHFWQZDJSROOH
|
7.7 | IC50 | 2 | — | |
JTVGTLWDQVRWPA
|
7.7 | IC50 | 2 | — | |
KBVKZTXBAARIBF
|
7.7 | IC50 | 2 | — | |
LMKUCXMEOPPASU
|
7.7 | IC50 | 2 | — | |
MEDCPPNEGZYFET
|
7.7 | IC50 | 2 | — | |
MLOCVODZBGTHFR
|
7.7 | IC50 | 2 | — | |
MSDDMDKQDPONFK
|
7.7 | IC50 | 2 | — | |
MYZDQYGTUAEWLQ
|
7.7 | IC50 | 2 | — | |
OKBJYZHLIFUWOD
|
7.7 | IC50 | 2 | — | |
QIUAPKYBHDKVCU
|
7.7 | IC50 | 2 | — | |
RNMYFUIDUIXUQF
|
7.7 | IC50 | 2 | — | |
RQLJMFJBLWRMIZ
|
7.7 | IC50 | 2 | — | |
RQQWCYPROZEXIC
|
7.7 | IC50 | 2 | — | |
UDDMNBYVRLYNKY
|
7.7 | IC50 | 2 | — | |
UDZJPUXBHJZZKD
|
7.7 | IC50 | 2 | — | |
VDZJXIOFISBBLT
|
7.7 | IC50 | 2 | — | |
WCEILCDOSWQPTH
|
7.7 | IC50 | 2 | — | |
WLMIPQKDBNGKKU
|
7.7 | IC50 | 2 | — | |
YMAMZOHSCXVQEM
|
7.7 | IC50 | 2 | — | |
ZGZUTVMOEPZIBL
|
7.7 | IC50 | 2 | — | |
AFUGPLVMIXYSOF
|
7.7 | IC50 | 2 | — | |
CZHJQAJYLJCDOF
|
7.7 | Ki | 2 | — |