Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZGQOYORTUCLRJE
|
7.9 | IC50 | 2 | — | |
ZRYHQJAOERFYMX
|
7.9 | IC50 | 2 | — | |
ZWDMOCLWOFLYJB
|
7.9 | IC50 | 2 | — | |
XRENHHRXIIBXTK
|
7.9 | IC50 | 2 | — | |
NJQQFMIMUJWYJW
|
7.9 | IC50 | 2 | — | |
SWKCNNNINQTNKE
|
7.9 | IC50 | 2 | — | |
YALKQTNPKCPCSL
|
7.9 | IC50 | 2 | — | |
AFMYOEOCOWXZLE
|
7.8 | IC50 | 2 | — | |
DZOQWZXXMIBPGC
|
7.8 | IC50 | 2 | — | |
KINBCVMCTUBHEP
|
7.8 | IC50 | 2 | — | |
LDKJJCMTYSYKGC
|
7.8 | IC50 | 2 | — | |
NOIQCRFIOYMHLK
|
7.8 | IC50 | 2 | — | |
RARAMGIQFJHXBX
|
7.8 | IC50 | 2 | — | |
YHMDEFKWDBLHED
|
7.8 | IC50 | 2 | — | |
MNZXPIGNPIOMFO
|
7.8 | IC50 | 2 | — | |
UDTVMTVICUTHFZ
|
7.8 | IC50 | 2 | — | |
FKDHVFZSRUETTG
|
7.8 | IC50 | 3 | — | |
OXSVGZCCNVYPAP
|
7.8 | IC50 | 2 | — | |
PHPHYTVUIHUSDY
|
7.8 | IC50 | 2 | — | |
QGTBEOWAAMLRRE
|
7.8 | IC50 | 2 | — | |
QHEVATMKWCXSFO
|
7.8 | IC50 | 2 | — | |
UFNIBOWMYFHXAH
|
7.8 | IC50 | 2 | — | |
USURLDWGSGIIKO
|
7.8 | IC50 | 2 | — | |
UBGUQYHIHIWAKK
|
7.8 | IC50 | 3 | — | |
BAWWCXDEGWTQQJ
|
7.8 | IC50 | 2 | — | |
IOVVYYZLKVPLRE
|
7.8 | IC50 | 2 | — | |
JAEOMAZCAGUYJH
|
7.8 | IC50 | 2 | — | |
KEKRHNKYGGKUCC
|
7.8 | IC50 | 2 | — | |
LEOYYWVJQQAFPQ
|
7.8 | IC50 | 2 | — | |
NVMGFILMSZYTHH
|
7.8 | IC50 | 2 | — | |
OHNWUOJIEMWYKF
|
7.8 | IC50 | 2 | — | |
PFGKQRWHIVJCSQ
|
7.8 | IC50 | 2 | — | |
PPVANHMVSXBKKT
|
7.8 | IC50 | 2 | — | |
RJMFXJIFMYWTIU
|
7.8 | IC50 | 2 | — | |
VUYDSDDKXXDVBD
|
7.8 | IC50 | 2 | — | |
ZEDAXOJVMVPUQI
|
7.8 | IC50 | 2 | — | |
HIDSAPKGYMGXHV
|
7.8 | IC50 | 2 | — | |
ICUMRVYQEMSBSV
|
7.8 | IC50 | 2 | — | |
MSZLRJMCIIYHJP
|
7.8 | IC50 | 2 | — | |
NIVASVQLFPNGLI
|
7.8 | IC50 | 2 | — | |
YQBMOACVJAYNDW
|
7.8 | IC50 | 2 | — | |
ZLRYZXMLGYXCBB
|
7.8 | IC50 | 2 | — | |
HXYXHOWEKCGYDL
|
7.8 | Ki | 2 | — | |
OAGVOXBBBCESFK
|
7.8 | IC50 | 2 | — | |
CCCFPQTVEOSXNO
|
7.8 | IC50 | 2 | — | |
GKFAGGGLMOZPIH
|
7.8 | IC50 | 2 | — | |
GRVLSUPSKVOUTB
|
7.8 | IC50 | 2 | — | |
KSAAUHMSLCPIEX
|
7.8 | IC50 | 2 | — | |
NGKSRKYOGVIJBP
|
7.8 | IC50 | 2 | — | |
OPZYOXDFGXITFX
|
7.8 | IC50 | 2 | — |