Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRDGLJHBGVYYFD
|
8.0 | IC50 | 2 | — | |
NZVLXDCDEXMPNK
|
8.0 | IC50 | 2 | — | |
QKUFWMIANNNGBO
|
8.0 | IC50 | 2 | — | |
QOOKVBVTEODITI
|
8.0 | IC50 | 2 | — | |
WCFKPIGECORAJL
|
8.0 | Kd | 2 | — | |
XZKWHOTXDXTUIM
|
8.0 | IC50 | 2 | — | |
YVVGGNNZPPNCKL
|
8.0 | IC50 | 2 | — | |
ZSURMFSLVLIXJU
|
8.0 | IC50 | 2 | — | |
ZWVXEDURRJDRFT
|
8.0 | IC50 | 2 | — | |
ATYKKTVKFKHXRG
|
8.0 | IC50 | 2 | — | |
YSWYRVDXDMUHMQ
|
7.9 | IC50 | 2 | — | |
BFDPYKZZCCNXHD
|
7.9 | IC50 | 2 | — | |
BKBNLEXXXSBYJC
|
7.9 | IC50 | 2 | — | |
FUCYSTKEKHXIGJ
|
7.9 | IC50 | 2 | — | |
FWLGBMIRXNXBIW
|
7.9 | IC50 | 2 | — | |
IFXOKMOGQXWOAG
|
7.9 | IC50 | 2 | — | |
KQVCAKJYDIYLPP
|
7.9 | IC50 | 2 | — | |
SNKPYTPMXOONSA
|
7.9 | IC50 | 2 | — | |
VQWNFBGVGJSEIS
|
7.9 | IC50 | 2 | — | |
XAPZYJFLCOBOIV
|
7.9 | IC50 | 2 | — | |
IRIOIFXUMMFCIQ
|
7.9 | IC50 | 2 | — | |
FHQCHOTUQBIXHY
|
7.9 | IC50 | 3 | — | |
NKPHEWJJTGPRSL
|
7.9 | IC50 | 2 | — | |
PURFEOGTUNSLNC
|
7.9 | IC50 | 2 | — | |
AFORIMWHFCNSQW
|
7.9 | IC50 | 2 | — | |
BHAIZVDZNJCJEY
|
7.9 | IC50 | 2 | — | |
BIYLUSQJNYBVKQ
|
7.9 | IC50 | 2 | — | |
BXKCPLKQZJHTRJ
|
7.9 | IC50 | 2 | — | |
DZOBIUPSYGTFNB
|
7.9 | IC50 | 2 | — | |
FBJWNSGVHRPEHX
|
7.9 | IC50 | 2 | — | |
FGDRRSSGFWLPIU
|
7.9 | IC50 | 2 | — | |
GAPCXEBBIQPWQE
|
7.9 | IC50 | 2 | — | |
HCPUMVKWEGUHSQ
|
7.9 | IC50 | 2 | — | |
HRGZUWRNXHICSA
|
7.9 | IC50 | 2 | — | |
IGIWAQXIWHOQBF
|
7.9 | IC50 | 2 | — | |
IUPKPDHRHMPCIW
|
7.9 | IC50 | 2 | — | |
KAPPVWDHYWKMCP
|
7.9 | IC50 | 2 | — | |
KUZQLRMCUVSRAC
|
7.9 | IC50 | 2 | — | |
NKNOERDGAOLMLO
|
7.9 | IC50 | 2 | — | |
OECGRWHBAZTUJY
|
7.9 | IC50 | 2 | — | |
PYGWGZALEOIKDF
|
7.9 | IC50 | 5 | — | |
QDNNECCKGHNPJH
|
7.9 | IC50 | 2 | — | |
QJVZNZJGIQXUNN
|
7.9 | IC50 | 2 | — | |
SFDZUXBOFCZNSX
|
7.9 | IC50 | 2 | — | |
SVZKFADYBNPPGB
|
7.9 | IC50 | 2 | — | |
VOCHUPYGKFNXTA
|
7.9 | IC50 | 2 | — | |
WYAVQIMQXVYOJD
|
7.9 | IC50 | 2 | — | |
XIPQAWQDZQGDAP
|
7.9 | IC50 | 2 | — | |
XNQLEUZDIJTWDV
|
7.9 | IC50 | 2 | — | |
YLBKDRAXARKXCP
|
7.9 | IC50 | 2 | — |