Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBEMIKYVMRKEJZ
|
8.1 | IC50 | 2 | — | |
IYYZTRFPNHSBBR
|
8.1 | IC50 | 2 | — | |
ICMMROMWLJCAMI
|
8.1 | IC50 | 2 | — | |
JITRDWUJQJEPRS
|
8.1 | IC50 | 2 | — | |
DRSFMMJLALGGQD
|
8.1 | IC50 | 2 | — | |
FJLACAPWUVBMDA
|
8.1 | Ki | 2 | — | |
HMYOYYAKSLLNNF
|
8.1 | IC50 | 2 | — | |
JSTRBBFHRKOOAS
|
8.1 | IC50 | 2 | — | |
QLMYSNOBOJVFPQ
|
8.1 | IC50 | 2 | — | |
RONSOUVGSPQFBT
|
8.1 | IC50 | 2 | — | |
RVKKYYGCYYMTCF
|
8.1 | IC50 | 2 | — | |
YSKHEIVCJQLEOT
|
8.1 | IC50 | 2 | — | |
NCDWDCAWJRKYEV
|
8.0 | IC50 | 2 | — | |
VAILRUBYKONNMR
|
8.0 | IC50 | 2 | — | |
XRWCMYGWXHGDLW
|
8.0 | IC50 | 2 | — | |
BNBHRFGMJAMOPS
|
8.0 | IC50 | 2 | — | |
IDGCMHSOMGZCJU
|
8.0 | IC50 | 2 | — | |
NFZPQSVNLVXUOS
|
8.0 | IC50 | 2 | — | |
WYJSWDJMPDRABG
|
8.0 | IC50 | 2 | — | |
AOSLCGQGWXABMG
|
8.0 | IC50 | 3 | — | |
ZPBMUWYVRPVKAM
|
8.0 | IC50 | 2 | — | |
AVHFITFFUBSKNU
|
8.0 | IC50 | 2 | — | |
BKOCKOZLSUDOBA
|
8.0 | IC50 | 2 | — | |
BLZZAJBLYALRNA
|
8.0 | IC50 | 2 | — | |
CYYXTKIISNGPGF
|
8.0 | IC50 | 2 | — | |
DZMYZUPNSMGTEY
|
8.0 | IC50 | 2 | — | |
HULWVKFKDFHZQG
|
8.0 | IC50 | 2 | — | |
JKZAHWOFWBFJNL
|
8.0 | IC50 | 2 | — | |
MCJWFYQBNIPBAD
|
8.0 | IC50 | 2 | — | |
MJRKVMJMSUHOAI
|
8.0 | IC50 | 2 | — | |
MNRCVDCRFODXQB
|
8.0 | IC50 | 2 | — | |
PKTDOGBMTZCKJY
|
8.0 | IC50 | 2 | — | |
PLEUHERUYNIDFX
|
8.0 | IC50 | 2 | — | |
SANCCSVGFPHWTN
|
8.0 | IC50 | 2 | — | |
TWHPGIQZGKDNQM
|
8.0 | IC50 | 2 | — | |
ULHPGVYPONETEM
|
8.0 | IC50 | 2 | — | |
VCFANMMZFZDTIY
|
8.0 | IC50 | 2 | — | |
XIIOAQCZRAHEDV
|
8.0 | IC50 | 2 | — | |
XMLWIZXKPYHVRK
|
8.0 | IC50 | 2 | — | |
XZDQPIYQIWBLNV
|
8.0 | IC50 | 2 | — | |
ZHCKHDSIOBSCSP
|
8.0 | IC50 | 3 | — | |
DFMGGAHVNBGTNP
|
8.0 | IC50 | 2 | — | |
OKDKQGCRSIBHSQ
|
8.0 | IC50 | 2 | — | |
CTTVIEYMZPRCCH
|
8.0 | IC50 | 2 | — | |
FMYUTKMVQXUAHS
|
8.0 | IC50 | 2 | — | |
RRHDSDOQUUHQGB
|
8.0 | IC50 | 2 | — | |
ARHVTCINCFVQFC
|
8.0 | IC50 | 2 | — | |
CIUYCGPZIOUMNU
|
8.0 | IC50 | 2 | — | |
HAMCSLXJGSVTTJ
|
8.0 | IC50 | 2 | — | |
JOXLHLUBKIVNIJ
|
8.0 | IC50 | 2 | — |