Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AAYAGLDVWRKOPN
|
8.2 | IC50 | 2 | — | |
ALLQDFMKVJMXSZ
|
8.2 | IC50 | 2 | — | |
DCRLONDGVUVHIO
|
8.2 | IC50 | 2 | — | |
DLYWQFUMFDBURV
|
8.2 | IC50 | 2 | — | |
GDGAUOBZPMXAIE
|
8.2 | IC50 | 2 | — | |
HHWIGJYKVRTBFJ
|
8.2 | IC50 | 2 | — | |
JAWVBARHNLTQNK
|
8.2 | IC50 | 2 | — | |
KLMNQDGJZUNXGC
|
8.2 | IC50 | 2 | — | |
PKICVKLKMOBLLB
|
8.2 | IC50 | 2 | — | |
PUMHDEZGCLMKIC
|
8.2 | IC50 | 2 | — | |
QWUKBBWNPIGBCU
|
8.2 | IC50 | 2 | — | |
RYAIGLAQMMFJFE
|
8.2 | IC50 | 2 | — | |
SULJAFUYBRGUCY
|
8.2 | IC50 | 2 | — | |
AIFBSHYMNHBOFH
|
8.2 | IC50 | 2 | — | |
FTUVUYXKBIUTBX
|
8.2 | IC50 | 2 | — | |
UVOJGEJSFVVDCT
|
8.2 | IC50 | 2 | — | |
IZLMIDCIDWPUFS
|
8.2 | IC50 | 2 | — | |
QXXQWIDOJKUBHN
|
8.2 | IC50 | 2 | — | |
RUUTXFMIBONPLT
|
8.2 | IC50 | 2 | — | |
AZARJASHNJUTBT
|
8.2 | IC50 | 2 | — | |
CKOJPIRIFOCJML
|
8.2 | IC50 | 2 | — | |
QGUAKBNBIUEYCD
|
8.2 | IC50 | 2 | — | |
KPACNXQOCFGJKO
|
8.2 | IC50 | 2 | — | |
RGDXKPQBVYZPLJ
|
8.2 | IC50 | 2 | — | |
BSORRSQYOBLMKM
|
8.2 | Ki | 2 | — | |
GYAFBLINDLEUJW
|
8.2 | IC50 | 2 | — | |
KNQKGLODDLNGTC
|
8.2 | IC50 | 2 | — | |
KPVDIIPFHYNTLD
|
8.2 | IC50 | 2 | — | |
PZCHTGMFZMPABI
|
8.2 | IC50 | 2 | — | |
SBUMXUSAHHKUBE
|
8.2 | IC50 | 2 | — | |
SWGDXLAZBZDUBR
|
8.2 | IC50 | 3 | — | |
VKQKEROEGYSHIY
|
8.2 | IC50 | 2 | — | |
GCSJGOQPSGYWLQ
|
8.1 | Ki | 2 | — | |
MBIDFEZSWRDKLB
|
8.1 | IC50 | 2 | — | |
YEFVOKDOLXVJEU
|
8.1 | IC50 | 2 | — | |
AVRQNXKPTRWLBE
|
8.1 | IC50 | 2 | — | |
HLMCQIOABIQLTH
|
8.1 | IC50 | 2 | — | |
SMIKEPVXNWPXRL
|
8.1 | IC50 | 2 | — | |
BMQKNCOLHCNITG
|
8.1 | IC50 | 2 | — | |
BVGFFMVYNQSJKW
|
8.1 | IC50 | 2 | — | |
IEZOLPNZJAVUST
|
8.1 | IC50 | 2 | — | |
IHCSNCPUXYAQOH
|
8.1 | IC50 | 2 | — | |
JDPBFYPOTBVWBU
|
8.1 | Ki | 2 | — | |
MCNQPZJFPCWMBX
|
8.1 | IC50 | 2 | — | |
URBRWOCTHYUBBB
|
8.1 | IC50 | 2 | — | |
WDYJSZQUBJOQCI
|
8.1 | IC50 | 2 | — | |
ZDQQNHIPLGUZCD
|
8.1 | IC50 | 2 | — | |
ZOPMUEQEVARESV
|
8.1 | IC50 | 2 | — | |
IGFYSEGGTKFZIF
|
8.1 | IC50 | 2 | — | |
SRXZTYXSCXTZAL
|
8.1 | IC50 | 2 | — |