Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OLZLESUYMWMOIH
|
8.4 | IC50 | 2 | — | |
OPOMYANLMWFFAL
|
8.4 | IC50 | 2 | — | |
UGXMERDWVUNBBX
|
8.4 | IC50 | 2 | — | |
VFQDFESUBBNARZ
|
8.4 | IC50 | 2 | — | |
VMZCSGVUCCGELW
|
8.4 | IC50 | 2 | — | |
YWRMGNFFDSLFNI
|
8.4 | IC50 | 2 | — | |
UBXXFDJETHMQAG
|
8.4 | IC50 | 2 | — | |
CUYHWBGVPXGMKQ
|
8.4 | Ki | 2 | — | |
PMVRLVXVFQPYOQ
|
8.4 | Ki | 2 | — | |
QAPCSQPQKODCBU
|
8.4 | Ki | 2 | — | |
YGWYLCTVXDISQZ
|
8.4 | IC50 | 2 | — | |
YZMDGUHXAPIFCJ
|
8.4 | IC50 | 2 | — | |
IQHOGIMNAWJGAN
|
8.4 | IC50 | 2 | — | |
UDDMCWWGJNYNIG
|
8.4 | IC50 | 2 | — | |
LFYBZBXUCNISLC
|
8.3 | IC50 | 2 | — | |
QOWQLJPKVFLTTM
|
8.3 | IC50 | 2 | — | |
QSAWJDNKFPMGBM
|
8.3 | Ki | 2 | — | |
CCCGMNJZPJSHEU
|
8.3 | IC50 | 2 | — | |
MGOSAGCMMBAHOF
|
8.3 | IC50 | 2 | — | |
FHPFSIJRJJGJIS
|
8.3 | IC50 | 2 | — | |
CFXNTAQVKSBORV
|
8.3 | IC50 | 2 | — | |
DIDKWCOCQJWMDJ
|
8.3 | IC50 | 3 | — | |
DPMNJGIGYUPXKX
|
8.3 | IC50 | 2 | — | |
DSKHTBOXJLSDKF
|
8.3 | IC50 | 3 | — | |
IZTWDVIZDRDIQB
|
8.3 | IC50 | 2 | — | |
JFIAVEATUHYZRN
|
8.3 | IC50 | 2 | — | |
JOHAYHVXYQNTLV
|
8.3 | IC50 | 2 | — | |
MEMZMTDLGYXQLT
|
8.3 | IC50 | 2 | — | |
MRMQXYKAPMAYOL
|
8.3 | IC50 | 2 | — | |
PGCWVKQUBZQNGJ
|
8.3 | IC50 | 2 | — | |
PZYJPOPJUOPKCU
|
8.3 | IC50 | 2 | — | |
QJPPUQKBYWSDLP
|
8.3 | IC50 | 2 | — | |
UDLNAIHPWDPZTR
|
8.3 | IC50 | 2 | — | |
WPGGQAPGDRZFDF
|
8.3 | IC50 | 2 | — | |
XBHXUZVSEVBCGV
|
8.3 | IC50 | 2 | — | |
ZFILMNZQPSHFSZ
|
8.3 | IC50 | 2 | — | |
ZZRRYEXYIVBDNM
|
8.3 | IC50 | 2 | — | |
VPPLBZFNSZPKNK
|
8.3 | IC50 | 2 | — | |
AVNBRYDGABAMIV
|
8.3 | Ki | 2 | — | |
HQGAUHGLDUZZOL
|
8.3 | IC50 | 2 | — | |
WXGVTZYUTNQLMV
|
8.3 | IC50 | 2 | — | |
YMZRHLSISUIVFY
|
8.3 | IC50 | 2 | — | |
BCZSPEANUSIVNQ
|
8.3 | IC50 | 2 | — | |
GRJOAOUKNDQSQZ
|
8.3 | IC50 | 2 | — | |
XIWJYQJWSFRHJL
|
8.3 | Ki | 2 | — | |
BXNBZWBCCYYYDM
|
8.2 | IC50 | 2 | — | |
IGRNPARNLSUQKX
|
8.2 | IC50 | 2 | — | |
DFVOHJVISHJIGD
|
8.2 | IC50 | 2 | — | |
NLSDACBTLSVVEY
|
8.2 | IC50 | 2 | — | |
QPPRISSDNAGMFK
|
8.2 | IC50 | 2 | — |