Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTOMIMSUTLPSHA
|
8.6 | IC50 | 2 | — | |
JFIAVEATUHYZRN
|
8.6 | IC50 | 2 | — | |
LPQYTOYTUGNTHQ
|
8.6 | IC50 | 2 | — | |
QQWLDKMLZHRQRI
|
8.6 | IC50 | 2 | — | |
GYBNBRVJAPRVLI
|
8.6 | IC50 | 2 | — | |
GCSGUSKCFDTWJA
|
8.6 | IC50 | 2 | — | |
HKMAYQXCIOLGBJ
|
8.5 | IC50 | 2 | — | |
ANVDAXBIMHWBRJ
|
8.5 | IC50 | 2 | — | |
AWAKIULNKVOBKE
|
8.5 | IC50 | 2 | — | |
BEQOWVUOJYDODX
|
8.5 | IC50 | 2 | — | |
BOOFKKBANNNNAY
|
8.5 | IC50 | 2 | — | |
CROHJOSBERFQRJ
|
8.5 | IC50 | 2 | — | |
FIASQQMTLFRFPZ
|
8.5 | IC50 | 2 | — | |
HHUZWDREJDTDKG
|
8.5 | IC50 | 2 | — | |
HSRURUKCXSZMPN
|
8.5 | IC50 | 2 | — | |
JHPFXXSFWCODRI
|
8.5 | IC50 | 2 | — | |
JYWCOSPTGRQYHC
|
8.5 | IC50 | 2 | — | |
MRFNXYCMJVBPGQ
|
8.5 | IC50 | 3 | — | |
OHQMEDBYNUAVNE
|
8.5 | IC50 | 2 | — | |
QPIYUHRAHJHMRR
|
8.5 | Ki | 2 | — | |
RDDOUZYTYQTOLV
|
8.5 | IC50 | 2 | — | |
RTMMFLXVQPUVNI
|
8.5 | Ki | 2 | — | |
TWHPGIQZGKDNQM
|
8.5 | IC50 | 2 | — | |
VGPRZMGEBOLDGA
|
8.5 | IC50 | 2 | — | |
WZTJXUAIMNGSNF
|
8.5 | IC50 | 2 | — | |
YQEKTGDIFUMXQN
|
8.5 | IC50 | 2 | — | |
ZOPLPSKLHFWWGT
|
8.5 | IC50 | 2 | — | |
MVKIBLGTARYSKO
|
8.5 | IC50 | 2 | — | |
ZLFJCZVDOSFNSI
|
8.5 | IC50 | 2 | — | |
QRLZBRIZBGLFAE
|
8.5 | IC50 | 2 | — | |
SQGNYTDBQSSZEE
|
8.5 | IC50 | 2 | — | |
REDZQXWKFVNPGL
|
8.5 | IC50 | 2 | — | |
YMRUCOCNLHJFRC
|
8.5 | Ki | 2 | — | |
DTCDDPOBJLMFDD
|
8.5 | IC50 | 2 | — | |
GCBABDNEHNSTQA
|
8.5 | IC50 | 2 | — | |
XNQLEUZDIJTWDV
|
8.5 | IC50 | 2 | — | |
JPSHATBRSXMHDD
|
8.4 | Ki | 2 | — | |
BMOJLYKWVNBRLY
|
8.4 | IC50 | 2 | — | |
SXELKXZIKMONBL
|
8.4 | Ki | 2 | — | |
HMOAABYAIGYFNW
|
8.4 | IC50 | 2 | — | |
JKGNOCZOVVBHFE
|
8.4 | IC50 | 2 | — | |
RVBDITSUSNBLOS
|
8.4 | IC50 | 2 | — | |
KKDFGWKNYMTGFQ
|
8.4 | IC50 | 2 | — | |
DGQCQEKWSKAFOT
|
8.4 | IC50 | 2 | — | |
BTAYUWNJKKALGC
|
8.4 | IC50 | 2 | — | |
FKUXHXTYZGJMGB
|
8.4 | IC50 | 2 | — | |
IPURPIAIQWFSPQ
|
8.4 | IC50 | 2 | — | |
JMAGRGYNUBAGRG
|
8.4 | IC50 | 2 | — | |
MBXVAZICFZAFMX
|
8.4 | IC50 | 2 | — | |
MKHQMHQQWORQTO
|
8.4 | IC50 | 2 | — |