Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEKLFDBRFNKVQJ
|
7.2 | IC50 | 2 | — | |
UDJDZBKDACDLLY
|
7.2 | IC50 | 2 | — | |
XLGMFHHPUVDLQD
|
7.2 | IC50 | 2 | — | |
HMFATUVSGNYXMG
|
7.2 | IC50 | 2 | — | |
PPBACBMUIDHVDG
|
7.2 | IC50 | 2 | — | |
SPQWDVLQSPPBAJ
|
7.2 | IC50 | 2 | — | |
ULZRRGUANDXXBI
|
7.2 | IC50 | 2 | — | |
WLXIJLBHOZKHSY
|
7.2 | IC50 | 2 | — | |
BPGJBCJVDGOSGO
|
7.2 | IC50 | 2 | — | |
CCJJPOCNADHZMF
|
7.2 | IC50 | 2 | — | |
CGZMGUYTVASJAL
|
7.2 | IC50 | 2 | — | |
CXEWRFDQZWGKCT
|
7.2 | IC50 | 2 | — | |
GNMFKYCBSKMWKN
|
7.2 | IC50 | 2 | — | |
HQXBICNDMZIHKY
|
7.2 | IC50 | 2 | — | |
IPVNHELRRJRWDT
|
7.2 | IC50 | 2 | — | |
IZCCLPQZOODGAE
|
7.2 | IC50 | 2 | — | |
KBEMBRRTXOGSLG
|
7.2 | IC50 | 2 | — | |
KLSNOFKRRAEBGB
|
7.2 | IC50 | 2 | — | |
KWWWAPRSFOPABI
|
7.2 | IC50 | 2 | — | |
NZDLBBJYDRLQCG
|
7.2 | IC50 | 2 | — | |
RNSYNDAURDULIZ
|
7.2 | IC50 | 2 | — | |
RUFQBYAUEBPVOC
|
7.2 | IC50 | 2 | — | |
ZHALZSRGISCBSZ
|
7.2 | IC50 | 2 | — | |
GYIOHTJWSJFTCV
|
7.2 | IC50 | 2 | — | |
KHJNUJLYIHQWQI
|
7.2 | IC50 | 3 | — | |
LQQHADUYCCSZCE
|
7.2 | IC50 | 2 | — | |
NEBHLBAEPITUDU
|
7.2 | IC50 | 2 | — | |
OJJVULINVLFCDX
|
7.2 | IC50 | 2 | — | |
BBMSVWIHGBXKOG
|
7.1 | IC50 | 2 | — | |
FCLSFIPJKQGFST
|
7.1 | IC50 | 2 | — | |
FKOIZIQMOBSDJT
|
7.1 | IC50 | 2 | — | |
HBLBBNLKFJMUIP
|
7.1 | IC50 | 2 | — | |
IOWSBZYCNNDVIQ
|
7.1 | IC50 | 2 | — | |
ISDVLXGUCZEBAA
|
7.1 | IC50 | 2 | — | |
LOSVSQZYWMNMOM
|
7.1 | IC50 | 2 | — | |
LUVBXQXGHNHXKY
|
7.1 | IC50 | 2 | — | |
OBLNEWAKNNXMEQ
|
7.1 | Ki | 2 | — | |
OFRPOQBLTULHQG
|
7.1 | IC50 | 2 | — | |
OPULJURKAOMYQN
|
7.1 | IC50 | 2 | — | |
PCISUPGLSWCBQO
|
7.1 | IC50 | 2 | — | |
SVODMOAKIUXEHE
|
7.1 | IC50 | 2 | — | |
XVZVVBATNVUIRX
|
7.1 | IC50 | 2 | — | |
ZWDMOCLWOFLYJB
|
7.1 | IC50 | 2 | — | |
ILVWSEURLCBURN
|
7.1 | IC50 | 2 | — | |
LSQBARLEVVWISB
|
7.1 | IC50 | 2 | — | |
WNKWNLLPIAKZAB
|
7.1 | IC50 | 2 | — | |
HLEGFMMPJFQDLU
|
7.1 | IC50 | 2 | — | |
INNRTYATIQKSRB
|
7.1 | IC50 | 2 | — | |
JLWXEFNEFHBDLL
|
7.1 | IC50 | 2 | — | |
PNXTVJPPVFEKCU
|
7.1 | IC50 | 2 | — |