Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCSTYDSAUMAZOK
|
7.2 | IC50 | 2 | — | |
NKKNLQBFWFWENA
|
7.2 | IC50 | 2 | — | |
OWQJVODOCWCIPX
|
7.2 | IC50 | 2 | — | |
QOQOEYLFCWZWJM
|
7.2 | IC50 | 2 | — | |
QSEZKNHRUQRMIL
|
7.2 | IC50 | 2 | — | |
VTWDQQNZHHCVKP
|
7.2 | IC50 | 2 | — | |
YHOYZBOLGRMWLY
|
7.2 | IC50 | 2 | — | |
DJTPMKUBCLTTCX
|
7.2 | IC50 | 2 | — | |
IEEKRCLQMYQEAW
|
7.2 | IC50 | 2 | — | |
MKWAVIYAYROLPX
|
7.2 | IC50 | 2 | — | |
AKFJHUREZCFDBB
|
7.2 | IC50 | 2 | — | |
BSMBUEWDJYQNBV
|
7.2 | IC50 | 2 | — | |
CSSYYMDTOQBMBE
|
7.2 | IC50 | 2 | — | |
HINMFTUIHCBZCY
|
7.2 | IC50 | 2 | — | |
JWDXFZMJSOKLBM
|
7.2 | IC50 | 2 | — | |
LIYNCRHQGJVEOI
|
7.2 | IC50 | 2 | — | |
MDUVTBXIIMXLNO
|
7.2 | IC50 | 2 | — | |
OQWSGTUKBXDUJN
|
7.2 | IC50 | 2 | — | |
QADWTEIFYFLHLO
|
7.2 | IC50 | 2 | — | |
QTFAFXQTVIFDBF
|
7.2 | IC50 | 2 | — | |
RBFYUIXVWQHOIR
|
7.2 | IC50 | 2 | — | |
RIPOGUPNVLZOCZ
|
7.2 | IC50 | 2 | — | |
ULVUURBFDYVMPY
|
7.2 | IC50 | 2 | — | |
XNKLLVCARDGLGL
|
7.2 | IC50 | 2 | — | |
YITDREASSSCOKM
|
7.2 | IC50 | 2 | — | |
ZLAVJBBRIDICHK
|
7.2 | IC50 | 2 | — | |
DRBRRJMHVFQSGA
|
7.2 | IC50 | 2 | — | |
MCVZDSBUIGAXFL
|
7.2 | IC50 | 2 | — | |
MLPJJJZFUUSHAR
|
7.2 | IC50 | 2 | — | |
OKQBAEDMKCFVFW
|
7.2 | IC50 | 2 | — | |
OTEQAQOANIBUPR
|
7.2 | IC50 | 2 | — | |
SJNMBQBKAJVHAR
|
7.2 | IC50 | 2 | — | |
YLSQNVPQNURPHL
|
7.2 | IC50 | 2 | — | |
YQXCVAGCMNFUMQ
|
7.2 | IC50 | 2 | — | |
BAWOOMZYWPDRIV
|
7.2 | IC50 | 2 | — | |
BKXUZQUTEZBQIW
|
7.2 | IC50 | 2 | — | |
ITLJTFLFDKESMH
|
7.2 | IC50 | 2 | — | |
QBVRPSNZXYJPPT
|
7.2 | IC50 | 2 | — | |
VYOWQMFTCPKETE
|
7.2 | Ki | 2 | — | |
AYCCBDPQSLELEH
|
7.2 | IC50 | 2 | — | |
DXQDLUHFSIHLID
|
7.2 | IC50 | 2 | — | |
DYSAONVHJLEPIL
|
7.2 | IC50 | 2 | — | |
KXBYACQQJJSRDU
|
7.2 | IC50 | 2 | — | |
LFPUYQWXIHQGCT
|
7.2 | IC50 | 2 | — | |
VLMFZDMYBOXYJH
|
7.2 | IC50 | 2 | — | |
WFNGFPISCALAAF
|
7.2 | IC50 | 2 | — | |
WZKHNVLGIMDJSQ
|
7.2 | IC50 | 2 | — | |
GOSIJUGDTWLDOF
|
7.2 | IC50 | 2 | — | |
LUYCFGBPBPYQHG
|
7.2 | IC50 | 2 | — | |
NJEZYJRDECMCSF
|
7.2 | IC50 | 2 | — |