Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LPBHCIIMBZNWQE
|
7.3 | IC50 | 2 | — | |
LRVAUDNAIRDUQD
|
7.3 | IC50 | 2 | — | |
ONJALOWSUSAVJN
|
7.3 | IC50 | 2 | — | |
QDMNPIRGCSJFLT
|
7.3 | IC50 | 2 | — | |
RHYOCTPUTIOWJU
|
7.3 | IC50 | 2 | — | |
SBNQDANULLAFPB
|
7.3 | IC50 | 2 | — | |
UMDZTWFRNJDGSH
|
7.3 | IC50 | 2 | — | |
UNKRRBWXJZNMAN
|
7.3 | IC50 | 2 | — | |
UQPHCFHWXAYPSB
|
7.3 | IC50 | 2 | — | |
WUKFGTRLGMGCPE
|
7.3 | IC50 | 2 | — | |
XDLNWPYQPUIONK
|
7.3 | IC50 | 2 | — | |
XERIEOGWOGJQKP
|
7.3 | IC50 | 2 | — | |
XGUKQJNTBMFLGV
|
7.3 | IC50 | 2 | — | |
MYCUZCCPKYVWHO
|
7.3 | IC50 | 2 | — | |
PSAZZQBVZAAEEQ
|
7.3 | IC50 | 2 | — | |
WIZBIQCUWVRTIO
|
7.3 | IC50 | 3 | — | |
BYNRVAUPJHWXBV
|
7.3 | IC50 | 2 | — | |
FLSSHCYZWNMCNZ
|
7.3 | IC50 | 2 | — | |
MAZUVMQRDUXXOS
|
7.3 | IC50 | 2 | — | |
PDGLHDNSYURVOE
|
7.3 | IC50 | 2 | — | |
UCRABRKSDLESNY
|
7.3 | IC50 | 2 | — | |
VBZNCCCGPNUSTO
|
7.3 | IC50 | 2 | — | |
XNKOXOVQENJNQC
|
7.3 | IC50 | 2 | — | |
ZOHWDHISAPBPKM
|
7.3 | IC50 | 2 | — | |
ALLWDYBEXBKRLB
|
7.3 | IC50 | 2 | — | |
PRXSJOIEHROIED
|
7.3 | IC50 | 2 | — | |
VNZUEWWSRMNKNI
|
7.3 | IC50 | 2 | — | |
ZKKPMROIYVDVAG
|
7.3 | IC50 | 2 | — | |
ZXZVCBMMKZOPKU
|
7.3 | IC50 | 2 | — | |
GISQDTWWOXOIKD
|
7.3 | IC50 | 2 | — | |
HASDKQMKEXOVJW
|
7.3 | IC50 | 2 | — | |
JRTBBYIREZFTKB
|
7.3 | IC50 | 2 | — | |
LIBNIJRKGCRKDJ
|
7.3 | IC50 | 2 | — | |
MGLVBVHKXIGSHJ
|
7.3 | IC50 | 2 | — | |
NTSXHAFEAVEPHI
|
7.3 | IC50 | 2 | — | |
WVVQRRCTXQZQNC
|
7.3 | IC50 | 2 | — | |
XGSPOMGPMJAGAH
|
7.3 | IC50 | 2 | — | |
XUIZIBCKVKBTGV
|
7.3 | Ki | 2 | — | |
AKWCEBKOJSOHOC
|
7.2 | IC50 | 2 | — | |
CCRFIOFFGAXDSM
|
7.2 | IC50 | 2 | — | |
KKRIIQWMMUVKTF
|
7.2 | IC50 | 2 | — | |
KPVRJZZBKQIDOC
|
7.2 | IC50 | 2 | — | |
LNEUEUNCOYSMKB
|
7.2 | IC50 | 2 | — | |
LNKZHPYDPHHQJV
|
7.2 | IC50 | 2 | — | |
QBVPZFQWBKTFNA
|
7.2 | IC50 | 2 | — | |
CSMNTPGYEWJYMN
|
7.2 | IC50 | 2 | — | |
CTQRTSFDXNIPBR
|
7.2 | IC50 | 2 | — | |
HQXBICNDMZIHKY
|
7.2 | IC50 | 2 | — | |
JCWXZLDZUNAWDL
|
7.2 | IC50 | 2 | — | |
JQEHHYUUNKMJPP
|
7.2 | IC50 | 2 | — |