Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LIZCIYFUFWQVAN
|
7.4 | IC50 | 2 | — | |
LJIMJRPXJPGBAF
|
7.4 | IC50 | 2 | — | |
NVZCDOLEPUQGGF
|
7.4 | IC50 | 2 | — | |
QPRGKOPOCKMWTN
|
7.4 | IC50 | 2 | — | |
QZOGWNOXUZLRLL
|
7.4 | IC50 | 2 | — | |
LHKJZFNHQDGATR
|
7.4 | IC50 | 2 | — | |
ULVQHUJNLXHURY
|
7.4 | IC50 | 2 | — | |
ZBYMCOLWOMSHIN
|
7.4 | IC50 | 2 | — | |
ZIAOVIPSKUPPQW
|
7.4 | IC50 | 2 | — | |
AQHMBDAHQGYLIU
|
7.3 | IC50 | 4 | — | |
FHJGAWQBOVTBCY
|
7.3 | IC50 | 2 | — | |
IGBORPMTTHEACU
|
7.3 | IC50 | 2 | — | |
JEUJSDKSNPDSPD
|
7.3 | Ki | 2 | — | |
SXLRVUYLYFNPIP
|
7.3 | IC50 | 2 | — | |
UKMJJMHWYKEQMZ
|
7.3 | IC50 | 2 | — | |
UPBLRJDHIONRBX
|
7.3 | IC50 | 2 | — | |
ZALINBUDHHHXOE
|
7.3 | IC50 | 2 | — | |
CLEYUGQORIJGAS
|
7.3 | IC50 | 2 | — | |
DGBVNIAUNCJNBL
|
7.3 | IC50 | 2 | — | |
GSGCCRKJFOBKKU
|
7.3 | IC50 | 2 | — | |
MFDKEHDMGROWDJ
|
7.3 | IC50 | 2 | — | |
PSJAXWANWSDNBE
|
7.3 | IC50 | 2 | — | |
QELZVZAEUOTTEF
|
7.3 | IC50 | 2 | — | |
QHUTWTQVWQWDHJ
|
7.3 | IC50 | 2 | — | |
QVFQRVFKTQRRSW
|
7.3 | IC50 | 2 | — | |
UZQLDBWLAOCBOO
|
7.3 | IC50 | 2 | — | |
UZQLDBWLAOCBOO
|
7.3 | IC50 | 3 | — | |
XSPCPGMXRMWJOO
|
7.3 | IC50 | 2 | — | |
HBDRPGIVGNPAHP
|
7.3 | IC50 | 2 | — | |
HRZCTRGNLVWTGP
|
7.3 | IC50 | 2 | — | |
WOULWISOHTZRJX
|
7.3 | IC50 | 2 | — | |
XIDVTNDDDXQJCF
|
7.3 | IC50 | 2 | — | |
YAHRSQPSOHWRFW
|
7.3 | IC50 | 2 | — | |
FOHQBRBSZDTCTF
|
7.3 | IC50 | 2 | — | |
IECRVRWMRCHCKJ
|
7.3 | IC50 | 2 | — | |
MJPLPIUGKOHVQU
|
7.3 | IC50 | 2 | — | |
QKALTFMJVRCJEX
|
7.3 | IC50 | 2 | — | |
FIJHLQUEDUYOLI
|
7.3 | IC50 | 2 | — | |
HCYAKUPQJAVYPS
|
7.3 | IC50 | 2 | — | |
JKEVDPUWXLGMPH
|
7.3 | IC50 | 2 | — | |
KMSOGCRKDIIWQW
|
7.3 | IC50 | 2 | — | |
ADRUSCXPXYBGLP
|
7.3 | IC50 | 2 | — | |
CPXSCMDBZJDCCN
|
7.3 | Ki | 2 | — | |
DQAHTOGPWKESEP
|
7.3 | IC50 | 2 | — | |
GENVKPWACMTLDQ
|
7.3 | IC50 | 2 | — | |
HQXBICNDMZIHKY
|
7.3 | IC50 | 2 | — | |
JSZPCWCYYSOCKA
|
7.3 | IC50 | 2 | — | |
JYDIPPPAHISWJQ
|
7.3 | IC50 | 2 | — | |
JZEXVASPUCGEGB
|
7.3 | IC50 | 2 | — | |
LFYWPMJWZMLUDM
|
7.3 | IC50 | 2 | — |