Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VIKCADRKXGMLKS
|
7.4 | IC50 | 2 | — | |
WJBQILBCHRFMQR
|
7.4 | IC50 | 2 | — | |
XWIOCCJHKJBFSD
|
7.4 | IC50 | 2 | — | |
FHLDQZZHWVOPOC
|
7.4 | IC50 | 2 | — | |
SKROTKCZEQBLNS
|
7.4 | IC50 | 2 | — | |
SZJUURXLLYTLKS
|
7.4 | Ki | 2 | — | |
WUEBMTNCIUQAAC
|
7.4 | IC50 | 2 | — | |
GSLBQKHXBYDHEM
|
7.4 | IC50 | 2 | — | |
UPKYAAANFCQHRK
|
7.4 | IC50 | 2 | — | |
VIKLGGPFTSLKCS
|
7.4 | IC50 | 2 | — | |
WIAHHWDLCXFARH
|
7.4 | IC50 | 2 | — | |
ZSVRWYQPXDWCBM
|
7.4 | IC50 | 2 | — | |
AXDQTVHZYRQIIQ
|
7.4 | IC50 | 2 | — | |
CQFHTAOWHQBLSP
|
7.4 | Ki | 2 | — | |
JFMKEUCKWUZCOC
|
7.4 | IC50 | 2 | — | |
UIGJYHSYHVEEOI
|
7.4 | IC50 | 2 | — | |
YWFCIRVBIKEMHQ
|
7.4 | IC50 | 2 | — | |
BIKSKZHGVCCQDN
|
7.4 | IC50 | 2 | — | |
IIWLQNGPKWAHDD
|
7.4 | IC50 | 3 | — | |
ITIVZMJXVUFETB
|
7.4 | IC50 | 2 | — | |
JMHMFMJZTZPCBL
|
7.4 | IC50 | 2 | — | |
KXFVFUYEOVDVGN
|
7.4 | IC50 | 2 | — | |
MMHIUSFCQUDMTN
|
7.4 | IC50 | 2 | — | |
MRSDMFHPBHPUME
|
7.4 | IC50 | 2 | — | |
NRYKUUUTSXXIGZ
|
7.4 | IC50 | 2 | — | |
OSEJQKRMCRXNGM
|
7.4 | IC50 | 2 | — | |
POZPQWWKQDWCKE
|
7.4 | IC50 | 3 | — | |
QODMNQLSDFVBJL
|
7.4 | IC50 | 2 | — | |
QVBCGVSBAZFFCX
|
7.4 | IC50 | 2 | — | |
RLBNGNODRRYBOJ
|
7.4 | IC50 | 2 | — | |
VQJKUVSKZOTZTB
|
7.4 | Ki | 2 | — | |
WOULWISOHTZRJX
|
7.4 | IC50 | 2 | — | |
WYZVEMYGCLUVLS
|
7.4 | IC50 | 2 | — | |
XFTCXYNSTYIUTL
|
7.4 | IC50 | 2 | — | |
YDFFSHCXESSOAN
|
7.4 | IC50 | 2 | — | |
YHKPRNMRRSYRRC
|
7.4 | IC50 | 2 | — | |
LUTJEKVTRXUUAW
|
7.4 | IC50 | 2 | — | |
ZWDMOCLWOFLYJB
|
7.4 | IC50 | 2 | — | |
IWPVGRJQBHHROO
|
7.4 | IC50 | 2 | — | |
MWEQHXSWZIUDPO
|
7.4 | IC50 | 2 | — | |
NFHRPWYBGVVVMV
|
7.4 | IC50 | 2 | — | |
NGEDNFKTVIOWEY
|
7.4 | IC50 | 2 | — | |
NYOYRWHDZQWRFQ
|
7.4 | IC50 | 2 | — | |
QPWFFPQWSFQAFJ
|
7.4 | IC50 | 2 | — | |
UQMLJOLGLHVTER
|
7.4 | IC50 | 2 | — | |
UXRFRQBRUGBAOV
|
7.4 | IC50 | 2 | — | |
VTPUXUOCJGFEIT
|
7.4 | IC50 | 2 | — | |
DLUINPJNECTRBI
|
7.4 | IC50 | 2 | — | |
JUECZHWXFHYUAT
|
7.4 | IC50 | 2 | — | |
KGWRKSLKDXAWRK
|
7.4 | IC50 | 2 | — |