Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTYHXCRYMXKNCE
|
7.5 | IC50 | 2 | — | |
KCCUCWCDLCVQBS
|
7.5 | IC50 | 2 | — | |
KKDXAEVIBXHCBE
|
7.5 | IC50 | 2 | — | |
LOYHBPLQFXFEPV
|
7.5 | IC50 | 2 | — | |
LSDYBXHTYOZVST
|
7.5 | IC50 | 2 | — | |
NIINQTIUVDCATJ
|
7.5 | IC50 | 2 | — | |
OSCVHOFAXPMNHC
|
7.5 | IC50 | 2 | — | |
RGHSEODWAAUYRU
|
7.5 | IC50 | 2 | — | |
SSBDRFPTUIJDHD
|
7.5 | IC50 | 2 | — | |
XPOQHMRABVBWPR
|
7.5 | IC50 | 5 | — | |
YCNRDJWVQRPBNZ
|
7.5 | IC50 | 2 | — | |
YVMOAVJHQOOGCA
|
7.5 | IC50 | 2 | — | |
ZUVVXYGGMSOHJK
|
7.5 | Ki | 2 | — | |
JJWJSIAJLBEMEN
|
7.5 | IC50 | 3 | — | |
JMMPZYQZVRRZDH
|
7.5 | IC50 | 2 | — | |
NSMWIFFOQGJUCP
|
7.5 | IC50 | 2 | — | |
SVNKYELSAOAWPV
|
7.5 | IC50 | 2 | — | |
WFJSRRPSTPATRH
|
7.5 | IC50 | 2 | — | |
YXBIKCUVUPTBKE
|
7.5 | IC50 | 2 | — | |
ACDHMYCDBLZDSM
|
7.5 | IC50 | 2 | — | |
IDKAQKKABQCPDY
|
7.5 | IC50 | 2 | — | |
KVAKNJULNOOMID
|
7.5 | IC50 | 2 | — | |
LSOMQLHUCGDDFP
|
7.5 | IC50 | 2 | — | |
OFZPTYFLZZXCJA
|
7.5 | IC50 | 2 | — | |
RYMXRFRWLPSTHP
|
7.5 | IC50 | 2 | — | |
ZOSPYFFFYNDONY
|
7.5 | IC50 | 2 | — | |
FQVDJZWFSZSGGA
|
7.5 | IC50 | 2 | — | |
KRRNTBCBBOEWDQ
|
7.5 | IC50 | 2 | — | |
CLSMMEOPBVDYIA
|
7.5 | IC50 | 2 | — | |
GHRLOSINCJHBPV
|
7.5 | IC50 | 2 | — | |
GQMFTUBBCVWGHH
|
7.5 | IC50 | 2 | — | |
UCPAUURHWRDVKU
|
7.5 | IC50 | 2 | — | |
XPQJLGCHNKJKLR
|
7.5 | IC50 | 2 | — | |
DCTURVKYYUBBDN
|
7.5 | IC50 | 2 | — | |
PQYRXENYFNNRKX
|
7.5 | IC50 | 2 | — | |
PVONVQAXGDZBJO
|
7.5 | IC50 | 2 | — | |
QLRFOQAJDSEUSU
|
7.5 | IC50 | 2 | — | |
SZFTVMMXACFMSI
|
7.5 | IC50 | 2 | — | |
UUNRTTUYSMGSQR
|
7.5 | IC50 | 2 | — | |
VPIPMVMIKZKSSD
|
7.5 | IC50 | 2 | — | |
WXZWCTNRPUWZPF
|
7.5 | IC50 | 2 | — | |
HDVZWQWXAQRFKJ
|
7.5 | IC50 | 3 | — | |
QNDVBRRFKQCCLW
|
7.5 | Ki | 2 | — | |
SJGIKNOOIMIQBF
|
7.5 | IC50 | 2 | — | |
SNZLKNMCCWNHEG
|
7.5 | IC50 | 2 | — | |
TYPYIAOCHCKFIA
|
7.5 | IC50 | 2 | — | |
LIFRUTHXRYPBGV
|
7.4 | IC50 | 2 | — | |
MYZWNPZPNUEKQC
|
7.4 | IC50 | 2 | — | |
SGXGPYTZBKLAIU
|
7.4 | IC50 | 2 | — | |
URKZMNUSADOUAO
|
7.4 | IC50 | 2 | — |