Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HZXTYUBDPUXDNV
|
7.6 | IC50 | 2 | — | |
LHJSBTOSBYRXRM
|
7.6 | IC50 | 2 | — | |
MKYVJXCFWCUGQQ
|
7.6 | IC50 | 2 | — | |
RMXYGIHJODGJHN
|
7.6 | IC50 | 2 | — | |
XGBUEAAOXNGUJL
|
7.6 | IC50 | 2 | — | |
XGULEBRNTWJUHP
|
7.6 | IC50 | 2 | — | |
RBGHMPUVQIWMCT
|
7.6 | IC50 | 2 | — | |
HINKPOQANFSSAS
|
7.6 | IC50 | 2 | — | |
IDDNPJCCIQGGIR
|
7.6 | IC50 | 2 | — | |
MAUXHCDRJBNVBB
|
7.6 | IC50 | 2 | — | |
NTUKAXBBRWLMRL
|
7.6 | IC50 | 2 | — | |
QUJVYRZJKYTIDQ
|
7.6 | IC50 | 2 | — | |
RWKNTTWVISWZLP
|
7.6 | IC50 | 2 | — | |
UWBOVNUZRAIRLM
|
7.6 | IC50 | 2 | — | |
WDGALFMNQDRWDS
|
7.6 | IC50 | 2 | — | |
YIFNEVZKJSHELK
|
7.6 | IC50 | 2 | — | |
YPGBGYIRJKQKPA
|
7.6 | IC50 | 2 | — | |
DZMMOIFXNAEIHX
|
7.6 | IC50 | 2 | — | |
FWLIJFLHZVSBOP
|
7.6 | IC50 | 2 | — | |
HPKRLZZAMUMBAN
|
7.6 | IC50 | 2 | — | |
LBBBEFUIIOQXAR
|
7.6 | IC50 | 2 | — | |
LNEJMGHEKJARHP
|
7.6 | IC50 | 2 | — | |
OPPVYMRCOSOQGC
|
7.6 | IC50 | 2 | — | |
SVFUFLWHAVXRLA
|
7.6 | IC50 | 2 | — | |
UYUIJOAWTJMMIV
|
7.6 | IC50 | 2 | — | |
ABGHEVXZRVAYSV
|
7.5 | IC50 | 2 | — | |
HDOCGJCVEXCJAE
|
7.5 | Ki | 2 | — | |
IGHDGSYPBBTGNR
|
7.5 | IC50 | 2 | — | |
KWOXBTQBZVHKED
|
7.5 | IC50 | 2 | — | |
NPPGPCZJIKXPNW
|
7.5 | IC50 | 2 | — | |
SXPOHHRAMKMEHU
|
7.5 | IC50 | 3 | — | |
VTDODEQREQSSAV
|
7.5 | IC50 | 3 | — | |
XKSPCHATHZHOGY
|
7.5 | IC50 | 2 | — | |
BWLYGOVEEHWYDU
|
7.5 | IC50 | 2 | — | |
IVRVASYPWHAIIN
|
7.5 | IC50 | 2 | — | |
JWSYHRYRAITBIX
|
7.5 | IC50 | 2 | — | |
KBNAVAPRJRYDCX
|
7.5 | IC50 | 2 | — | |
OACOGSCQKYRDSY
|
7.5 | IC50 | 2 | — | |
XEHZKPPJHGBGNP
|
7.5 | Ki | 2 | — | |
IIIWVJXRUFDJEN
|
7.5 | IC50 | 2 | — | |
AETWZMHUXWRPAH
|
7.5 | IC50 | 2 | — | |
CHBMGMAGCOPBHF
|
7.5 | IC50 | 2 | — | |
CHUHSBRSLSCCSX
|
7.5 | IC50 | 3 | — | |
DCXXRUXBIXIQKD
|
7.5 | IC50 | 2 | — | |
DUNMXVXAKKVRJV
|
7.5 | IC50 | 2 | — | |
DZAUZGQGZFBFOY
|
7.5 | IC50 | 2 | — | |
FTLVKPIQAUANGB
|
7.5 | IC50 | 2 | — | |
HEJZGGFJHZQHRW
|
7.5 | IC50 | 2 | — | |
HRXHKHXJYOIYON
|
7.5 | IC50 | 2 | — | |
IZZVAMWPYNONCO
|
7.5 | IC50 | 2 | — |