Target Details
| UniProt AC | Q72547 |
|---|---|
| Gene Symbol | pol |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00075 (RNase_H) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) |
Summary
- Multi-target molecules 1,888
- Clinical molecules 0
- Avg pChEMBL 7.09
Top Co-occurrence Targets
- reverse transcriptase 988 shared
- gag-pol 499 shared
- gag-pol 259 shared
- reverse transcriptase 143 shared
- 22 shared
- PPIA 18 shared
- KCNH2 5 shared
- FEN1 4 shared
- ERCC5 3 shared
- TRM3 3 shared
Active Molecules (1,888)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZVNNERAAYHFPD
|
9.7 | IC50 | 2 | — | |
SVMHTBVIPYVDIL
|
9.7 | IC50 | 2 | — | |
KXDIHAQCVNNLIB
|
9.4 | IC50 | 2 | — | |
QWNIWQCTNAQHAF
|
9.4 | Ki | 2 | — | |
AASLKIYYTISYOA
|
9.3 | Ki | 2 | — | |
RURQSSZVFHRLEE
|
9.3 | Ki | 2 | — | |
UMHXETHRMTWBPR
|
9.3 | Ki | 2 | — | |
PRHGIYDCDMLXHN
|
9.3 | IC50 | 2 | — | |
FZBAOOQVQXATRL
|
9.2 | Ki | 2 | — | |
IOUDUHWREIAEKP
|
9.2 | IC50 | 2 | — | |
JWDAEHXXNUMMKQ
|
9.2 | Ki | 2 | — | |
AOIKBWIBFXPPRC
|
9.1 | IC50 | 2 | — | |
RXQSMZOUOHXYOX
|
9.1 | IC50 | 2 | — | |
ATXSRWHPTOHHAY
|
9.0 | IC50 | 2 | — | |
FLGARVIJXJZDND
|
9.0 | IC50 | 2 | — | |
GUSPHNVTAWXCCQ
|
9.0 | IC50 | 2 | — | |
PCUWRGFJGCYISU
|
9.0 | IC50 | 2 | — | |
TWONRKIIQCCNQJ
|
9.0 | IC50 | 2 | — | |
UOZDWSRONYZLQO
|
9.0 | IC50 | 2 | — | |
USWKTQVAABDFSY
|
9.0 | IC50 | 2 | — | |
YQELPLJAHMWKIX
|
9.0 | Ki | 2 | — | |
NPXCVIODFSNHMU
|
9.0 | IC50 | 2 | — | |
POOBUACLMWERDQ
|
9.0 | IC50 | 2 | — | |
UMPSTPLBACSCDI
|
9.0 | IC50 | 2 | — | |
GCZMATZWHYCJTH
|
8.9 | IC50 | 2 | — | |
BFPBNKBYNOBOHM
|
8.9 | IC50 | 2 | — | |
NKPHEWJJTGPRSL
|
8.9 | Kd | 2 | — | |
ZSDYTNJSFLYICM
|
8.9 | Ki | 2 | — | |
BUECGHMIFPUORL
|
8.9 | IC50 | 2 | — | |
WHCLIFOVZDANCU
|
8.9 | IC50 | 2 | — | |
ABOZXYNAPFTBHX
|
8.8 | Ki | 2 | — | |
SBDZLPIXOSPFIW
|
8.8 | IC50 | 2 | — | |
UUVBMMWJHPNLHN
|
8.8 | IC50 | 2 | — | |
IJTWXTIWZPKVDV
|
8.8 | IC50 | 2 | — | |
NTNSGKOURZQJSK
|
8.8 | IC50 | 2 | — | |
OCABMICVVJLNTB
|
8.8 | Ki | 2 | — | |
PNJKKJNQGSBNDN
|
8.8 | IC50 | 2 | — | |
SSFUYPBGOTXADP
|
8.8 | IC50 | 2 | — | |
RUEZUQUJOIHYNQ
|
8.8 | Ki | 2 | — | |
YCIPBZALVAZULV
|
8.7 | Ki | 2 | — | |
DNNXGKQZFKHVRU
|
8.7 | IC50 | 2 | — | |
IDNIWMWKAMOXLP
|
8.7 | IC50 | 2 | — | |
KVJCKKKSJAZIHH
|
8.7 | IC50 | 2 | — | |
NZABYUMWKMPSBX
|
8.7 | IC50 | 2 | — | |
SZLMFNKKFJUHKQ
|
8.7 | IC50 | 2 | — | |
SSUZBIFUDPSYGO
|
8.7 | IC50 | 2 | — | |
JNNYBFVTFNQISB
|
8.7 | IC50 | 2 | — | |
RGRSOJUFXZMIHM
|
8.7 | IC50 | 2 | — | |
PJDCZSKXLVBCNA
|
8.6 | Ki | 2 | — | |
USRHSVZSPKDGMT
|
8.6 | IC50 | 2 | — |