Target Details
UniProt ACQ70Z44
Gene SymbolHTR3D
Protein Name5-hydroxytryptamine receptor 3D
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 182
  • Clinical molecules 6
  • Avg pChEMBL 7.85
Top Co-occurrence Targets
Active Molecules (182)
InChIKey pChEMBL Type Targets Clinical
SGKHROGKIKKECN 7.6 Ki 5
XQMDXRYDYUXFEH 7.5 Ki 5
YVTHPCKJOKJJHA 7.5 IC50 5
FEPRMAUTVAUZGM 7.5 IC50 5
VQMVUGKLGFORBP 7.5 IC50 5
LWLBVIFUVSUSAY 7.5 Ki 6
DWLMIHRZURMFAQ 7.5 Ki 5
KIJXVALDJPUIFM 7.5 Ki 6
LDIYRDXQPDSEFR 7.5 IC50 5
HASGWVOTHYCRIP 7.4 Ki 5
KIVOPFOXJNXWFW 7.4 Ki 5
OOMBBUZQJGYRRW 7.4 Ki 5
FCZBQMUDGBEIHG 7.4 Ki 5
JZSPAHAWDCQCEX 7.4 Ki 5
DAZOPYDOJHNKSD 7.4 Ki 5
NWVOTDQIZMJKRJ 7.4 Ki 5
SDFWQNVGYRAAAZ 7.3 Ki 5
FMWXWOAWFBYPCO 7.3 IC50 5
BMIQQALNTAJMLB 7.3 Ki 5
SSOHJAKQLOENEM 7.3 Ki 6
TTWJBBZEZQICBI 7.3 Kd 10
JXOLMXLINBXECI 7.3 Ki 5
UMHNYWDDWJWNHJ 7.2 Kd 5
GGDBEAVVGFNWIA 7.2 Ki 6
XFRTZUYXJVAJNT 7.2 Ki 5
MKWFJPZMYHPQIA 7.2 Ki 5
VHFVKMTVMIZMIK 7.2 Ki 15
HMOMXYPGOQVVIY 7.2 Kd 5
LGKSUDPSBCMQRR 7.2 Ki 5
XQJMXPAEFMWDOZ 7.2 Kd 5
XOUOEUATRAFRCX 7.2 Ki 5
HNDKJDCYXITJAR 7.2 Ki 5
GIRLVGYIIVFTLI 7.1 Ki 6
ZSTKHSQDNIGFLM 7.1 Kd 22
DEMZYMHKNNMIGU 7.1 IC50 5
PXAINPSPSFFTMA 7.1 IC50 5
WPVVMKYQOMJPIN 7.0 Ki 5
DCSUBABJRXZOMT 7.0 Kd 24
ARCIIEQRTPPAQU 6.9 IC50 5
PDTVBRINWYWWLT 6.9 Ki 5
QZAYGJVTTNCVMB 6.9 Ki 17
AXKDMCQUCRBQFP 6.8 Ki 5
GAYSOZKZPOVDSB 6.8 Ki 5
VNICFCQJUVFULD 6.8 Ki 15
AFLJKKMTBWNZFE 6.7 Ki 6
HKPHVFFQXHMOHX 6.7 Ki 5
KVWDHTXUZHCGIO 6.7 Ki 32 Yes
ZXTPPBDZBKAHMV 6.7 Kd 5
HTYFFCPFVMJTKM 6.7 Ki 5
BRNUKIDBYPCLGD 6.7 IC50 5
2D structure