Target Details
| UniProt AC | Q6XUX3 |
|---|---|
| Gene Symbol | DSTYK |
| Protein Name | Dual serine/threonine and tyrosine protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 14
- Clinical molecules 5
- Avg pChEMBL 6.53
Associated Diseases (2)
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
QQWUGDVOUVUTOY
|
7.2 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
UBPYILGKFZZVDX
|
6.4 | Kd | 130 | Yes | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
MFAQYJIYDMLAIM
|
6.3 | Kd | 130 | Yes | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
DSKYHEJWWIBREA
|
6.2 | Kd | 8 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
JRNJNYBQQYBCLE
|
6.1 | Kd | 40 | Yes | |
CTNPALGJUAXMMC
|
6.0 | Kd | 151 | — |