Target Details
| UniProt AC | Q6V1X1 |
|---|---|
| Gene Symbol | DPP8 |
| Protein Name | Dipeptidyl peptidase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF19520 (Dpp_8_9_N) PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 337
- Clinical molecules 0
- Avg pChEMBL 7.16
Active Molecules (337)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKYQMUOQXBQKOO
|
7.0 | IC50 | 3 | — | |
YCHHGVIQSNZGAO
|
7.0 | Ki | 3 | — | |
YCHHGVIQSNZGAO
|
7.0 | Ki | 3 | — | |
TUHONCVWZIUJQF
|
6.9 | IC50 | 3 | — | |
DKOFRISURGKKQT
|
6.9 | IC50 | 2 | — | |
JUTVQMDQVZFLGD
|
6.9 | IC50 | 3 | — | |
UBDCHKXSBGAGNJ
|
6.9 | IC50 | 2 | — | |
XGNBIYXILDDDQR
|
6.9 | IC50 | 4 | — | |
CUQPRCWWJPLANH
|
6.9 | IC50 | 2 | — | |
HXSMSCXZJMHYRH
|
6.9 | IC50 | 3 | — | |
GBAHBSLKOOONMN
|
6.9 | IC50 | 2 | — | |
ZEMFLZQUUHJMGT
|
6.9 | IC50 | 6 | — | |
RYWOUVPMSNURME
|
6.8 | Ki | 3 | — | |
JWANCNBNXTWMNU
|
6.8 | Ki | 2 | — | |
YDYSCRZHYWLSPQ
|
6.8 | IC50 | 2 | — | |
DYSZJGFBTWPUEV
|
6.8 | Ki | 5 | — | |
OOTQGBQMGZXPSV
|
6.8 | Ki | 4 | — | |
MMZVCOZOFNZWBM
|
6.8 | IC50 | 2 | — | |
CSYRDDZULSVTOA
|
6.8 | Ki | 2 | — | |
BXWYQMPOVCJLIS
|
6.8 | IC50 | 4 | — | |
MEGNCLBXJMSXAB
|
6.8 | IC50 | 2 | — | |
QAAMJGGJVHEAAE
|
6.8 | IC50 | 2 | — | |
DNQFYDFLXGMRRF
|
6.8 | IC50 | 2 | — | |
HJMXMWNMTNQTDK
|
6.8 | IC50 | 2 | — | |
DPVYMNCQRPIQEA
|
6.7 | IC50 | 3 | — | |
JBPNPLREHXKRHY
|
6.7 | IC50 | 3 | — | |
YWWWYGQQSBBBEZ
|
6.7 | Ki | 5 | — | |
CIYSGOBBUFBQIH
|
6.7 | IC50 | 3 | — | |
FFVYIARXOOWGNK
|
6.7 | IC50 | 2 | — | |
IJFVLVWFCVPKBM
|
6.7 | Ki | 2 | — | |
NRUIYKIBILMTRY
|
6.7 | IC50 | 2 | — | |
MAIFOHYNLBAWDL
|
6.7 | IC50 | 3 | — | |
YDVBKYKVTWRKIY
|
6.7 | IC50 | 3 | — | |
MKJRNYHUGVCOAT
|
6.7 | IC50 | 3 | — | |
NRTUDFQDPVFTRM
|
6.7 | IC50 | 2 | — | |
QLNACVPURHNJCY
|
6.7 | IC50 | 2 | — | |
VWKRRCNHGXGMJQ
|
6.7 | IC50 | 2 | — | |
WCRLBFHWFPELKW
|
6.7 | IC50 | 3 | — | |
WCRLBFHWFPELKW
|
6.7 | IC50 | 3 | — | |
UUKCXASWMAQVLX
|
6.6 | Ki | 3 | — | |
VDIQELAZMIFVDS
|
6.6 | Ki | 3 | — | |
DGFODDFZJTVDBE
|
6.6 | IC50 | 3 | — | |
MEPRZPLBMXAVKQ
|
6.6 | IC50 | 3 | — | |
MTBATCJDNBSLTB
|
6.6 | IC50 | 4 | — | |
NEGWJHQAWQAHOF
|
6.6 | Ki | 5 | — | |
QGJUIPDUBHWZPV
|
6.6 | IC50 | 3 | — | |
QKCRGRBXMIWGEO
|
6.6 | Ki | 4 | — | |
WAVJGCCRPYAHLF
|
6.6 | IC50 | 4 | — | |
SHQGMGKBRGBIGM
|
6.6 | IC50 | 4 | — | |
UZZDZARFWLTODD
|
6.6 | IC50 | 5 | — |