Target Details
| UniProt AC | Q6UW60 |
|---|---|
| Gene Symbol | PCSK4 |
| Protein Name | Proprotein convertase subtilisin/kexin type 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01483 (P_proprotein) PF00082 (Peptidase_S8) PF16470 (S8_pro-domain) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.22
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHSWXCHUJHYZLB
|
6.4 | Ki | 4 | — | |
XIHRZTWKTVFWSV
|
6.4 | Ki | 4 | — | |
GREDJTIKEQWSJW
|
6.3 | Ki | 4 | — | |
RYVHKZGUULZSGD
|
6.3 | Ki | 4 | — | |
ALKYWGCWYLWWQX
|
6.2 | Ki | 4 | — | |
ICMPUUKPBRMOSD
|
6.2 | Ki | 4 | — | |
GBWNVGJPAAAKFV
|
6.2 | Ki | 3 | — | |
GHIUMDOROBFONL
|
6.2 | Ki | 3 | — | |
BEXKWEWEAXISEC
|
6.1 | Ki | 3 | — | |
SPILXWOFMWMUJL
|
6.1 | Ki | 3 | — | |
ANHXASYJLDAVKI
|
6.0 | Ki | 4 | — |