Target Details
| UniProt AC | Q6S4W0 |
|---|---|
| Gene Symbol | CDPK1 |
| Protein Name | Calcium-dependent protein kinase 1 |
| Organism | Cryptosporidium parvum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 88
- Clinical molecules 3
- Avg pChEMBL 8.03
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FDHLEBRUJJZXMR
|
8.1 | IC50 | 2 | — | |
VTPYDZCVVYWSRL
|
8.1 | IC50 | 2 | — | |
IIGJAOIYTPPGAN
|
8.1 | IC50 | 2 | — | |
LJDXURUFAXNINU
|
8.1 | IC50 | 2 | — | |
MMRLNUFECMEMSQ
|
8.1 | IC50 | 3 | — | |
VINBTOORIXBXPF
|
8.1 | IC50 | 2 | — | |
QNWAWMYUVHCJOJ
|
8.0 | IC50 | 2 | — | |
MZPILEJBIWMIFA
|
7.9 | IC50 | 3 | — | |
GCJVZJWLFLYCJR
|
7.9 | IC50 | 2 | — | |
UZRSJQXLFKNVMY
|
7.9 | IC50 | 2 | — | |
ZCXUCDWNAIZDKS
|
7.9 | IC50 | 2 | — | |
BLUGXYZMSPGIAA
|
7.8 | IC50 | 2 | — | |
VZGULHBHJBIHDH
|
7.8 | IC50 | 2 | — | |
AMGMAKSGXBFINM
|
7.7 | IC50 | 2 | — | |
CPIBWXJDDLOQSC
|
7.7 | IC50 | 2 | — | |
HGALDAPNHYJZAJ
|
7.7 | IC50 | 11 | Yes | |
VUSWSOVTPRKZMU
|
7.7 | IC50 | 2 | — | |
WBDAGEMKPQGVJA
|
7.7 | IC50 | 2 | — | |
SHQJMIVAJKVTPY
|
7.5 | IC50 | 2 | — | |
NLZUZMDQCFLSME
|
7.5 | IC50 | 4 | — | |
DKEXUOIKEUTIAL
|
7.5 | IC50 | 3 | — | |
XLHSLEFSSSWIGF
|
7.5 | IC50 | 3 | — | |
GSEFRQXISXMBJX
|
7.3 | IC50 | 2 | — | |
LKNZTNVERDBXML
|
7.3 | IC50 | 2 | — | |
OTWGEGUQDHMDBA
|
7.2 | IC50 | 3 | — | |
QIXQTQFKKYRSSM
|
7.2 | IC50 | 2 | — | |
JSONRPFPVGYCOB
|
7.1 | IC50 | 3 | — | |
QUPSOTTWHXSAPW
|
7.1 | IC50 | 2 | — | |
HGAJCAYHMBFUDT
|
7.0 | IC50 | 3 | — | |
LCQAIZAFSOZWRC
|
7.0 | IC50 | 8 | Yes | |
MCKFAQNBWBWWAZ
|
6.9 | IC50 | 2 | — | |
TYDGXGDYKRIRIF
|
6.9 | IC50 | 3 | — | |
HMRUGEAVJFRORJ
|
6.8 | IC50 | 3 | — | |
NWHWDCQGLSTCCC
|
6.8 | IC50 | 2 | — | |
NWHSGEQUBWPLBD
|
6.7 | IC50 | 2 | — | |
BBTFPYWNKYLKIS
|
6.4 | IC50 | 2 | — | |
SZRCRQLPOHAVJL
|
6.4 | IC50 | 3 | — | |
XMTAJCWZZMFYID
|
6.2 | IC50 | 3 | — |