Target Details
| UniProt AC | Q6S4W0 |
|---|---|
| Gene Symbol | CDPK1 |
| Protein Name | Calcium-dependent protein kinase 1 |
| Organism | Cryptosporidium parvum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 88
- Clinical molecules 3
- Avg pChEMBL 8.03
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PTVXXUDFVRRVAE
|
9.4 | IC50 | 3 | — | |
NRRBFJRUKPITFY
|
9.2 | IC50 | 5 | — | |
ALIRNZFSPVRFPC
|
9.1 | IC50 | 3 | — | |
BRIJSCVHXQTNKX
|
9.0 | IC50 | 2 | — | |
KONPIFGGWNMOKY
|
9.0 | IC50 | 4 | — | |
XZLFLNWUBLMFQW
|
9.0 | IC50 | 2 | — | |
CMVANALWKBATOM
|
8.7 | IC50 | 2 | — | |
ONQFGFIAOHMNST
|
8.7 | IC50 | 2 | — | |
RLCOKRNYALYJSA
|
8.7 | IC50 | 2 | — | |
SVSZSOYWPORIAV
|
8.7 | IC50 | 2 | — | |
RUMXSJCIUQZQHF
|
8.7 | IC50 | 3 | — | |
CSXUIGRDFNAIAL
|
8.7 | IC50 | 3 | — | |
MBHHJCMRPHUOAD
|
8.6 | IC50 | 4 | — | |
ATIDQUUZAPHKND
|
8.5 | IC50 | 2 | — | |
LMHOKWLCLYLTHX
|
8.5 | IC50 | 2 | — | |
NUFMUAKSLVYPQF
|
8.5 | IC50 | 2 | — | |
OICIQHXOTTYPMV
|
8.5 | IC50 | 2 | — | |
RLTAZJWBDYRQHS
|
8.5 | IC50 | 2 | — | |
SPUWUOGLPPVXCW
|
8.5 | IC50 | 15 | Yes | |
WFGZCBMYRMUNLE
|
8.5 | IC50 | 2 | — | |
WGMMYAIGNLJDIM
|
8.5 | IC50 | 2 | — | |
YNCBHKFEHYLGFT
|
8.5 | IC50 | 2 | — | |
YTPFAWUHOBXMNJ
|
8.5 | IC50 | 2 | — | |
DLMBMHOJKBPKLK
|
8.5 | IC50 | 5 | — | |
DSVSFNREXPNTFM
|
8.4 | IC50 | 2 | — | |
ILMARQUWIMHOSG
|
8.4 | IC50 | 2 | — | |
ISFDEYBYSUBPMR
|
8.4 | IC50 | 2 | — | |
KKVWPXTXOCRUQG
|
8.4 | IC50 | 2 | — | |
QETVBRLPQMGMBP
|
8.4 | IC50 | 2 | — | |
BEHMFFDBKCHBHU
|
8.3 | IC50 | 2 | — | |
CKYKSFPZSGEXCP
|
8.3 | IC50 | 2 | — | |
IYNLAGHSNARNHP
|
8.3 | IC50 | 2 | — | |
JAEQFFFYQGMWDD
|
8.3 | IC50 | 2 | — | |
JDHOKTPTMDNUCI
|
8.3 | IC50 | 2 | — | |
JNCYMMFOKVMRMU
|
8.3 | IC50 | 2 | — | |
MXVDOTDIJVYNLE
|
8.3 | IC50 | 2 | — | |
NIWCEFPYEYYQMN
|
8.3 | IC50 | 2 | — | |
NPQIPWMDLIWSMO
|
8.3 | IC50 | 2 | — | |
QDNYKPYYLWQMPU
|
8.3 | IC50 | 2 | — | |
SOBPJJCTFHUZHH
|
8.3 | IC50 | 2 | — | |
XOYALPHJTHBLCG
|
8.3 | IC50 | 2 | — | |
YTSDNPLOCDVGNB
|
8.3 | IC50 | 8 | — | |
YXEUOWLDWIHNLO
|
8.3 | IC50 | 2 | — | |
JZGIKAAUVCHJDT
|
8.2 | IC50 | 2 | — | |
QHBDRDRJQJTZOX
|
8.2 | IC50 | 2 | — | |
XIGBSBUACNWRMJ
|
8.2 | IC50 | 2 | — | |
ZAQLYTILMDGYCM
|
8.2 | IC50 | 2 | — | |
ZJDQCUMJDLLUFT
|
8.2 | IC50 | 2 | — | |
YXMBIJKVPSHQMB
|
8.2 | IC50 | 2 | — | |
AJQKERUGIYLYDN
|
8.1 | IC50 | 2 | — |