Target Details
| UniProt AC | Q6PHR2 |
|---|---|
| Gene Symbol | ULK3 |
| Protein Name | Serine/threonine-protein kinase ULK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF04212 (MIT) PF00069 (Pkinase) |
Summary
- Multi-target molecules 35
- Clinical molecules 11
- Avg pChEMBL 6.85
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.9 | IC50 | 408 | — | |
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
NHHQJBCNYHBUSI
|
8.2 | Kd | 220 | — | |
QQWUGDVOUVUTOY
|
8.0 | Kd | 231 | Yes | |
OSVUGUHRKMMBSE
|
7.8 | Kd | 170 | — | |
NXSJMRCTGYTSTK
|
7.8 | Kd | 200 | — | |
RYYNGWLOYLRZLK
|
7.7 | Kd | 45 | — | |
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
CTNPALGJUAXMMC
|
7.4 | Kd | 151 | — | |
WINHZLLDWRZWRT
|
7.4 | Kd | 201 | Yes | |
LOLPPWBBNUVNQZ
|
7.3 | Kd | 97 | Yes | |
ODPGGGTTYSGTGO
|
7.2 | Kd | 153 | — | |
XZXHXSATPCNXJR
|
7.2 | Kd | 165 | Yes | |
KOZFSFOOLUUIGY
|
7.0 | Kd | 88 | Yes | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
PIQCTGMSNWUMAF
|
6.8 | Kd | 137 | Yes | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
GCIKSSRWRFVXBI
|
6.5 | Kd | 109 | Yes | |
MHPBLCYPFBBOND
|
6.5 | IC50 | 6 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
UBPYILGKFZZVDX
|
6.3 | Kd | 130 | Yes | |
BLQYVHBZHAISJM
|
6.3 | Kd | 21 | Yes | |
DKZYXHCYPUVGAF
|
6.3 | Kd | 112 | — | |
ALKJNCZNEOTEMP
|
6.3 | Kd | 55 | — | |
FLBNLJLONKAPLR
|
6.2 | Kd | 31 | — | |
AYCPARAPKDAOEN
|
6.2 | Kd | 73 | — | |
RITAVMQDGBJQJZ
|
6.2 | Kd | 43 | — | |
YOVVNQKCSKSHKT
|
6.1 | Kd | 15 | — | |
GUBJNPWVIUFSTR
|
6.0 | Kd | 103 | — | |
AAKJLRGGTJKAMG
|
6.0 | Kd | 50 | Yes | |
FFPHMUIGESPOTK
|
6.0 | IC50 | 6 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |