Target Details
| UniProt AC | Q6P3R8 |
|---|---|
| Gene Symbol | NEK5 |
| Protein Name | Serine/threonine-protein kinase Nek5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 9
- Clinical molecules 1
- Avg pChEMBL 6.46
Active Molecules (9)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHHQJBCNYHBUSI
|
7.9 | Kd | 220 | — | |
HKSZLNNOFSGOKW
|
7.0 | IC50 | 408 | — | |
ATWJOSDBVRWRHS
|
6.9 | IC50 | 5 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
HKSZLNNOFSGOKW
|
6.1 | Kd | 213 | — | |
VAARYSWULJUGST
|
6.0 | Kd | 119 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |