Target Details
UniProt ACQ6P179
Gene SymbolERAP2
Protein NameEndoplasmic reticulum aminopeptidase 2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF11838 (ERAP1_C) PF01433 (Peptidase_M1) PF17900 (Peptidase_M1_N)
Summary
  • Multi-target molecules 51
  • Clinical molecules 0
  • Avg pChEMBL 6.68
Top Co-occurrence Targets
Active Molecules (51)
InChIKey pChEMBL Type Targets Clinical
VCCACZUFRCVVFN 8.4 IC50 2
QKFOTLXPIIESQI 8.0 IC50 5
QHHKXYPPDICVAU 7.7 IC50 2
XAZJLAPNVJOSFR 7.5 IC50 2
FLHXMLUIEURZLV 7.4 IC50 3
QCPJTEUURKCRNT 7.4 IC50 4
SAZVKYFGANAWRA 7.3 IC50 3
JEQPENJEYBAHIE 7.2 IC50 3
GSWUIYHGTPVQDP 7.1 IC50 3
QJVIFKMCLOJOGV 7.1 IC50 3
AZIAPQRBCIAHTO 7.0 IC50 2
KAKJFMITKIMUAY 7.0 IC50 2
BUDSAEMPVYFKML 7.0 IC50 3
AATVMVZMTDKRJI 6.9 IC50 3
WVARWRXWGWJNRJ 6.9 IC50 3
PAISIGRMLVYIDB 6.9 IC50 3
WWNSEAAJQAYPMS 6.9 IC50 2
NJCHEVDWMWFDNQ 6.8 IC50 3
YSYQXQQIKOEBNN 6.8 Ki 3
MRXHFZNHXQEPNB 6.7 Ki 3
YNFZCLOZANIMIN 6.7 IC50 3
LWRKOPLMYMXZKW 6.7 Ki 2
BUDSAEMPVYFKML 6.7 IC50 2
WWZWLDVQUBJSGD 6.7 IC50 3
IEYYHWFOJFXPGP 6.7 IC50 3
SXZZIOOVCGCZRP 6.6 Ki 2
KFHOCODEDHRRMQ 6.6 IC50 2
ZGOYLLCQBCBXHF 6.6 IC50 3
ASBAZJSDHGVMRZ 6.5 IC50 3
QELOIXSGJMIHBZ 6.5 Ki 3
QELOIXSGJMIHBZ 6.5 Ki 4
FDAGDZVCWKCEEX 6.4 IC50 2
XFZZDIHCNHYESF 6.4 IC50 3
BUSBNAUESVLLQC 6.4 IC50 3
QELONQVCEFPRGM 6.3 IC50 2
JECKMXQKZJERLG 6.3 IC50 2
BEWRVZZHISITDQ 6.3 IC50 3
BEWRVZZHISITDQ 6.2 IC50 3
YHYCZFIGZSESIE 6.2 IC50 2
ZPHQKYQWQLYSDS 6.2 IC50 3
APTWADNFJQRAKY 6.2 IC50 2
GXEDNWSUKCJLLB 6.2 IC50 3
JREUTUCRLBCPNH 6.2 Ki 2
LCOBAHRSJLHENC 6.2 IC50 2
HUKAXHQRFRZFBN 6.1 IC50 2
WXYVFLSKRTUFAE 6.1 IC50 2
FWFGIHPGRQZWIW 6.1 IC50 6
LWNJKRUKVSPFJT 6.1 IC50 2
YNFZCLOZANIMIN 6.1 IC50 2
QWLYILUODIZPOK 6.0 IC50 3
2D structure